Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4016 |
BMS-986020
AM152,BMS986020 |
LPA Receptor; LPL Receptor | GPCR/G Protein |
BMS-986020 (AM152) 是一种高亲和力溶血磷脂酸受体 1 拮抗剂,有用于特发性肺纤维化的研究潜力。它抑制胆汁酸和磷脂转运蛋白,抑制 BSEP、MRP4 和 MDR3,IC50值分别为 4.8、6.2 和 7.5 μM。 | |||
TP1146 |
Adrenomedullin (AM) (1-52), human
Human adrenomedullin-(1-52)-NH2 |
||
Adrenomedullin (AM) (1-52), human is a 52-amino acid peptide that modulates cellular proliferation and angiogenesis in cancer. | |||
TP1145 |
Adrenomedullin (AM) (1-52), human TFA
Human adrenomedullin-(1-52)-NH2 (TFA) |
||
Adrenomedullin (AM) (1-52), human (TFA) is an NH2 terminal truncated adrenomedullin analogue,affects cell proliferation and angiogenesis in cancer. |