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Cat. No. Product Name Target Signaling Pathways
T16557 PNU-159682

Topoisomerase DNA Damage/DNA Repair
PNU-159682 是蒽环类新霉素的代谢产物,是一种 DNA 拓扑异构酶 II 抑制剂,具有出色的细胞毒性。
T4677 MMAD

Monomethylauristatin D,Demethyldolastatin 10,单甲基澳瑞他汀 D,Monomethyl Dolastatin 10

Microtubule Associated Cytoskeletal Signaling
MMAD (Demethyldolastatin 10) 是一种有效的微管蛋白抑制剂,是抗体药物偶联物中的一种毒素有效载荷。
T40879 7-MAD-MDCPT

7-MAD-MDCPT, a Camptothecin analog, is a toxin payload in antibody drug conjugates (ADCs).
T40872 17-AEP-GA

17-AEP-GA is a highly effective HSP90 antagonist compound that exhibits potent inhibition against the proliferation, survival, migration, and invasion of glioblastoma cells. Additionally, it demonstrates ADCs Toxin activity.
T11117 Duocarmycin MB

Others Others
Duocarmycin MB can be used against multi-drug resistant cell lines. Duocarmycin MB is an antibody drug conjugates (ADCs) toxin. Duocarmycin is a DNA alkylating agent that binds in the minor groove.
T11116 Duocarmycin MA

Others Others
Duocarmycin MA can be used against multi-drug resistant cell lines.Duocarmycin MA is an antibody drug conjugates (ADCs) toxin. Duocarmycin is a DNA alkylating agent that binds in the minor groove.
T10700 (+)-CBI-CDPI1

Others Others
(+)-CBI-CDPI1 is an enhanced functional analog of CC-1065. It is a DNA alkylating agent and an antibody-drug conjugates (ADCs) toxin.
T73948 Duocarmycin DM

Duocarmycin DM,一种DNA小沟烷基化剂(DNA minor-groove alkylator),作为抗体活性分子结合物(ADCs)的毒素,因其独特结构显示出抗癌活性。
T75117 Py-MAA-Val-Cit-PAB-DX8951

Py-MAA-Val-Cit-PAB-DX8951 是一种参与合成抗体药物偶联物(ADCs)中间体的嘌呤毒素。

化合物

PNU-159682
Cat.No: T16557
Synonym:
Target: Topoisomerase
MMAD
Cat.No: T4677
Synonym: Monomethylauristatin D,Demethyldolastatin 10,单甲基澳瑞他汀 D,Monomethyl Dolastatin 10
Target: Microtubule Associated
7-MAD-MDCPT
Cat.No: T40879
Synonym:
Target:
17-AEP-GA
Cat.No: T40872
Synonym:
Target:
Duocarmycin MB
Cat.No: T11117
Synonym:
Target: Others
Duocarmycin MA
Cat.No: T11116
Synonym:
Target: Others
(+)-CBI-CDPI1
Cat.No: T10700
Synonym:
Target: Others
Duocarmycin DM
Cat.No: T73948
Synonym:
Target:
Py-MAA-Val-Cit-PAB-DX8951
Cat.No: T75117
Synonym:
Target:
TargetMol Loading
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