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Cat. No. Product Name Target Signaling Pathways
T3024 Avitinib

AC0010,艾维替尼

EGFR; JAK; BTK Angiogenesis; Chromatin/Epigenetic; JAK/STAT signaling; Stem Cells; Tyrosine Kinase/Adaptors
Avitinib (AC0010) 是一种不可逆的、突变体选择性的EGFR 抑制剂,可有效抑制非小细胞肺癌中EGFR T790M 耐药突变。阿比替尼也是一种新型BTK 抑制剂。
T3721 Avitinib maleate

艾维替尼马来酸盐,艾维替尼

EGFR Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors
Avitinib maleate 是基于吡咯并嘧啶的不可逆的表皮生长因子受体抑制剂,IC50值为7.68 nM。
T70445 Lurtotecan dihydrochloride

Lurtotecan dihydrochloride is an antineoplastic (DNA Topoisomerase I Inhibitor)
T70446 Abivertinib HCl

Abivertinib, also known as AC0010 and Avitinib, is a third-generation EGFR tyrosine kinase inhibitor and BTK Inhibitor that demonstrated clinical efficacy and manageable adverse events (AEs). Abivertinib inhibits cell proliferation, reduces colony-forming capacity, and induces apoptosis and cell cycle arrest in AML cells, especially those harboring FLT3-ITD mutations. Abivertinib was also found to be more sensitive than ibrutinib in treating AML. Abivertinib may be a promising novel agent for A...

化合物

Avitinib
Cat.No: T3024
Synonym: AC0010,艾维替尼
Target: EGFR, JAK, BTK
Avitinib maleate
Cat.No: T3721
Synonym: 艾维替尼马来酸盐,艾维替尼
Target: EGFR
Lurtotecan dihydrochloride
Cat.No: T70445
Synonym:
Target:
Abivertinib HCl
Cat.No: T70446
Synonym:
Target:
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