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Cat. No. Product Name Target Signaling Pathways
T10213 A-437203

ABT-925,A37203,Lu201640

Dopamine Receptor GPCR/G Protein; Neuroscience
A-437203 (Lu201640) 是一种基于1H-pyrimidin-2-one scaffold 的、具有选择性的、新型强效的d3受体拮抗剂,对 D2, D3, 和 D4 受体,的Ki 值分别为 71, 1.6 和 6220 nM。
T69807 EGFR-IN-451

EGFR-IN-451 is an EGFR inhibitor, attenuating Ang II-induced Kidney Fibrosis.
T69808 ABT-925 fumarate

ABT-925, also known as A-37203, BSF-201640; DAT-201; Lu-201640; and A-437203, is a selective dopamine D3 receptor (DRD3) antagonist with an approximately 100-fold higher in vitro affinity for dopamine D₃ versus D₂ receptors. ABT-925 was tested in schizophrenia. ABT-925 is a selective dopamine D₃ receptor antagonist with an approximately 100-fold higher in vitro affinity for dopamine D₃ versus D₂ receptors.

化合物

A-437203
Cat.No: T10213
Synonym: ABT-925,A37203,Lu201640
Target: Dopamine Receptor
EGFR-IN-451
Cat.No: T69807
Synonym:
Target:
ABT-925 fumarate
Cat.No: T69808
Synonym:
Target:
TargetMol Loading
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