Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T2325 |
Neratinib
HKI-272,来那替尼 |
EGFR; HER | Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
Neratinib (HKI-272) 是一种口服的、不可逆的酪氨酸激酶抑制剂,对 HER2 和 EGFR 的 IC50值分别为 59 和 92 nM。 | |||
T71387 | Neratinib maleate monohydrate | ||
Neratinib maleate monohydrate is an irreversible inhibitor of the HER-2 receptor tyrosine kinase with potential antineoplastic activity. |