Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T61207 |
5-HT6/5-HT2A receptor ligand-1
|
||
5-HT6/5-HT2A receptor ligand-1 (compound 33) is a dual antagonist for the 5-HT6 and 5-HT2A receptors. It exhibits a K i value of 2 nM and 11 nM for the respective receptors. This compound holds promise for research in neurological and psychiatric disorders [1]. | |||
T61220 | 5-HT6/5-HT2A receptor ligand-2 | ||
5-HT6/5-HT2A receptor ligand-2 (化合物 42) 是一种可透过血脑屏障的5-HT6/5-HT2A 的双拮抗剂 ,Ki 值分别为 25 nM 和 32 nM。5-HT6/5-HT2A receptor ligand-2 具有促认知特性。 |