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Cat. No. Product Name Target Signaling Pathways
T1092 Zolmitriptan

佐米曲普坦,311C90,BW-311C90

5-HT Receptor GPCR/G Protein; Neuroscience
Zolmitriptan (311C90) 是一种5-HT1B/1D 受体部分激动剂,可用于偏头痛的研究,对 5-HT1B、5-HT1D、5-HT1F 受体的Ki 分别为 5.01、0.63 和 63.09 nM。
T0203 Sumatriptan succinate

舒马普坦琥珀酸盐,GR 43175,琥珀酸舒马曲坦

5-HT Receptor GPCR/G Protein; Neuroscience
Sumatriptan succinate (GR 43175) 是一种5-HT1受体激动剂,可作用于偏头疼的急性治疗。
T11326 Frovatriptan succinate hydrate

Frovelan,夫罗曲坦琥珀酸盐水合物 ,Frova

5-HT Receptor GPCR/G Protein; Neuroscience
Frovatriptan succinate hydrate (Frova) 是一种有效、高亲和力、选择性和口服活性的 5-HT1B、HT1D 受体激动剂和中等有效的 5-HT7 受体激动剂,pKi 值分别为 8.6、8.4 和 6.7。它可有效治疗各种偏头痛,包括恶心、呕吐、畏光和畏声等相关症状。
T1512 Rizatriptan benzoate

苯甲酸利扎曲坦,MK-462 Benzoate

5-HT Receptor GPCR/G Protein; Neuroscience
Rizatriptan benzoate (MK-462 Benzoate) 是 5-HT1激动剂,通过选择性结合并激活血清素 (5-HT) 1B 受体和 5-HT 1D 受体,从而缓解偏头痛。
T6602 Naratriptan hydrochloride

Naratriptan HCl,Amerge,Naramig,盐酸那拉曲坦,GR-85548A hydrochloride

5-HT Receptor GPCR/G Protein; Neuroscience
Naratriptan hydrochloride (GR-85548A hydrochloride) 是一种5-HT1受体激动剂,有抗偏头疼特性。它还可以通过刺激三叉神经系统感觉神经末梢上的 5-HT1D/1B 受体来发挥其作用,从而减少促炎神经肽的释放。
T60345 Frovatriptan

Frovatriptan is a highly potent agonist of the 5-HT 1B//D receptors, exhibiting the highest potency among triptan compounds. It possesses prominent cerebroselectivity. Frovatriptan demonstrates efficacy and even superiority in certain endpoints, including when administered during the headache phase of migraine attacks accompanied by aura [1].

化合物

Zolmitriptan
Cat.No: T1092
Synonym: 佐米曲普坦,311C90,BW-311C90
Target: 5-HT Receptor
Sumatriptan succinate
Cat.No: T0203
Synonym: 舒马普坦琥珀酸盐,GR 43175,琥珀酸舒马曲坦
Target: 5-HT Receptor
Frovatriptan succinate hydrate
Cat.No: T11326
Synonym: Frovelan,夫罗曲坦琥珀酸盐水合物 ,Frova
Target: 5-HT Receptor
Rizatriptan benzoate
Cat.No: T1512
Synonym: 苯甲酸利扎曲坦,MK-462 Benzoate
Target: 5-HT Receptor
Naratriptan hydrochloride
Cat.No: T6602
Synonym: Naratriptan HCl,Amerge,Naramig,盐酸那拉曲坦,GR-85548A hydrochloride
Target: 5-HT Receptor
Frovatriptan
Cat.No: T60345
Synonym:
Target:
TargetMol Loading
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