Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1600 |
Doxifluridine
Ro 21-9738,AMC 0101,5'-DFUR,5-Fluoro-5'-deoxyuridine,去氧氟尿苷 |
Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis | Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Doxifluridine (AMC 0101) 是一种胸苷磷酸化酶活化剂,对 PC9-DPE2细胞的 IC50为0.62 μM。它是具有抗肿瘤活性的抗肿瘤剂 5-fluorouracil (5-FU) 的氟嘧啶衍生物和口服前药。 | |||
TNU0621 |
5-Bromo-2’-fluoro-2’-deoxyuridine
|
||
Nucleoside, fluoro-modified nucleoside, halo-nucleoside | |||
T1408 |
Capecitabine
Xeloda,卡培他滨,Capecitibine,Capiibine,RO 09-1978 |
Apoptosis; Nucleoside Antimetabolite/Analog; DNA/RNA Synthesis | Apoptosis; Cell Cycle/Checkpoint; DNA Damage/DNA Repair |
Capecitabine (Capecitibine) 是一种可口服的前药,可由胸苷磷酸化酶催化转变为其活性代谢物 Fluorouracil。 |