Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TQ0002 |
A-317491
ABT 202 |
P2X Receptor | Membrane transporter/Ion channel; Neuroscience |
A-317491 (ABT 202) 是选择性和非核苷酸的 P2X3和 P2X2/3受体的拮抗剂,通过阻断 P2X3和 P2X2/3受体介导的钙通量减轻炎性和神经性疼痛。它对其他 P2 受体和神经递质受体,离子通道以及酶具有高度选择性,IC50大于10 μM。 | |||
T10204 |
A-317491 sodium salt hydrate
A-317491 sodium salt hydrate (475205-49-3 free base) |
Others | Others |
A-317491 sodium salt hydrate is a non-nucleotide P2X3 and P2X2/3 receptor antagonist, which inhibits calcium flux mediated by the receptors. |