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Cat. No. Product Name Target Signaling Pathways
T7465 4-Methylbenzylidene camphor

Enzacamene,4-甲基苄亚基樟脑,3-(4-甲基苯亚甲基)樟脑,4-MBC

AChE Neuroscience
4-Methylbenzylidene camphor 是有机的樟脑衍生物,应用于化妆品行业,具有保护皮肤抵抗紫外线(特别是紫外线B 辐射)的能力。
T0666 4-Chlorosalicylic acid

4-Chloro-2-hydroxybenzoic acid, 4-chloro salicylic acid,4-氯水杨酸

Tyrosinase; Antibacterial; Antibiotic; Antifungal Microbiology/Virology; Proteases/Proteasome
4-Chlorosalicylic acid (4-Chloro-2-hydroxybenzoic acid, 4-chloro salicylic acid) 是一种药物中间体。它抑制单酚酶和二苯酚酶活性,IC50值分别为1.89 mM 和1.10 mM。 它有抗菌活性,抑制大肠杆菌的MIC 为250 μg/mL,MBC 为500 μg/mL。
T36648 Tucatinib hemiethanolate

Tucatinib (Irbinitinib) hemiethanolate is a potent, orally active and selective HER2 inhibitor with an IC50 of 8 nM. Tucatinib hemiethanolate has nanomolar activity against purified HER2 enzyme and is approximately 500-fold selective for HER2 versus EGFR in cell-based assays. Tucatinib selectively inhibits the receptor tyrosine kinase HER2 relative to EGFR[1].Tucatinib blocks proliferation and the phosphorylation of HER2 and its downstream effector, Akt in HER2 overexpressing cell lines. In the ...

化合物

4-Methylbenzylidene camphor
Cat.No: T7465
Synonym: Enzacamene,4-甲基苄亚基樟脑,3-(4-甲基苯亚甲基)樟脑,4-MBC
Target: AChE
4-Chlorosalicylic acid
Cat.No: T0666
Synonym: 4-Chloro-2-hydroxybenzoic acid, 4-chloro salicylic acid,4-氯水杨酸
Target: Tyrosinase, Antibacterial, Antibiotic, Antifungal
Tucatinib hemiethanolate
Cat.No: T36648
Synonym:
Target:
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