Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T73128 | EGFR-IN-61 | EGFR | Angiogenesis; JAK/STAT signaling; Tyrosine Kinase/Adaptors |
EGFR-IN-61(化合物22a)为一种高效EGFR激酶抑制剂,其对L858R/T790M、L858R/T790M/C797S和WT的IC50值分别为42 nM、137 nM和743 nM。此外,EGFR-IN-61对A549和H1975细胞株展现抗增殖效应,其IC50值依次为2.14 μM和1.82 μM。 |