Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T9652 |
SB-747651A Dihydrochloride
|
ROCK | Cell Cycle/Checkpoint; Cytoskeletal Signaling; Stem Cells |
SB-747651A dihydrochloride是一种与ATP竞争性相互作用的抑制剂,特别针对丝裂原和应激激活激酶1 (MSK1),IC50值为11 nM。此化合物还能抑制PRK2、RSK1、p70S6K和ROCK-II等酶的活性。因其对上述激酶的抑制作用,SB-747651A dihydrochloride在炎症研究中显示出潜力。 | |||
T28695 |
SB-747651A
SB 747651A |
||
SB-747651A is a potent, ATP-competitive inhibitor of mitogen- and stress-activated kinase 1 (MSK1, IC50 = 11 nM). It targets the N-terminal kinase domain. SB-747651A inhibits MSK1, MSK2, PKA, PKB, RSK and p70S6K activity in cells. |