Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T16879 |
SHU 9119
|
Others | Others |
SHU 9119 is an effective human melanocortin 3 and 4 receptors (MC3/4R) antagonist and a partial MC5R agonist (IC50: 0.23, 0.06, and 0.09 nM for human MC3R, MC4R and MC5R, respectively). | |||
T16879L |
SHU 9119 acetate
SHU 9119 acetate (168482-23-3 free base) |
Melanocortin Receptor | GPCR/G Protein; Neuroscience |
SHU 9119 acetate 是众所周知的人黑皮质素 3 和 4 (hMC3R, hMC4R) 受体拮抗剂和部分 hMC5R 激动剂。人 MC3R、MC4R 和 MC5R 的 IC50 值分别为 0.23、0.06 和 0.09 nM。 |