Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7587 |
Tenapanor
RDX-5791,RDX 5791,AZD 1722,Tenapanor free base,RDX5791,AZD-1722,AZD1722 |
Sodium Channel | Membrane transporter/Ion channel |
Tenapanor (RDX 5791) 是钠氢离子交换NHE3的有效抑制剂, 对人和大鼠NHE3的IC50分别是5和10 nM。 | |||
T7587L |
Tenapanor HCl
RDX-5791,AZD 1722,AZD-1722,AZD1722,RDX5791,RDX 5791 |
||
Tenapanor( AZD-1722, RDX 5791) is an inhibitor of the sodium-proton (Na(+)/H(+)) exchanger NHE3, which is used for sodium handling in the gastrointestinal tract and kidney. |