Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4295 |
(R)-GNE-140
GNE-140 |
Dehydrogenase | Metabolism |
(R)-GNE-140 (GNE-140) 是 LDHA 抑制剂,能够作用于 LDHA (IC50:3 nM) 和 LDHB (IC50:3 nM)。它的活性是 S 型异构体的 18 倍。 | |||
T13450 | (S)-GNE-140 | Others | Others |
(S)-GNE-140 is the less active enantiomer of GNE-140. | |||
T13450L |
GNE-140 racemate
GNE-140 (racemate) |
Others | Others |
GNE-140 is a potent inhibitor of lactate dehydrogenase A (LDHA). GNE-140 is a racemate mixture of (R)-GNE-140 and (S)-GNE-140. | |||
T27421 |
GNE-140 racemic
GNE-140,GNE 140,GNE140 |
||
GNE-140 racemic is a potent lactate dehydrogenase (LDHA) inhibitor. |