Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T11139 |
(E/Z)-BCI
NSC 150117 |
Apoptosis; Phosphatase | Apoptosis; Metabolism |
(E/Z)-BCI (NSC-150117) 是一种DUSP6抑制剂,可通过激活 Nrf2 信号和抑制 NF-κB 通路,减弱 LPS 诱导的巨噬细胞炎症和 ROS 生成,具有抗炎活性。 | |||
T10486 |
BCI
(E)-BCI |
Phosphatase | Metabolism |
BCI ((E)-BCI) 是双重特异性磷酸酶的变构抑制剂。它特异性抑制 DUSP6和 DUSP1的 EC50分别为 13.3 和 8.0 μM,但不能够抑制 DUSP5。 | |||
T10486L |
BCI hydrochloride
(E)-BCI hydrochloride |
Others | Others |
BCI hydrochloride specifically inhibits DUSP6 and DUSP1 with EC50s of 13.3 and 8.0 μM in cells, respectively. BCI hydrochloride does not inhibit DUSP5. BCI hydrochloride is an allosteric inhibitor of dual specificity phosphatase (DUSP). |