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Cat. No. Product Name Target Signaling Pathways
T12480 Pipamperone

Floropipamide,McN-JR 3345,酰胺哌啶酮,R 3345

Others; Dopamine Receptor; 5-HT Receptor GPCR/G Protein; Neuroscience; Others
Pipamperone (McN-JR 3345) 是5-HT2A 受体和D4受体的高亲和力拮抗剂,也是D2受体的低亲和力拮抗剂,pKi 分别为 8.2、8.0 和 6.7。
T28417 Pipamperone HCl

fluoropipamide,floropipamide hydrochloride,carpiperone,floropipamide,R4050,Pipamperone

Pipamperone acts as an antagonist of the 5-HT2A, 5-HT2B, 5-HT2C D2, D3, D4, α1-adrenergic, and α2-adrenergic receptors. It shows much higher affinity for the 5-HT2A and D4 receptors over the D2 receptor (15-fold in the case of the D4 receptor, and even hi

化合物

Pipamperone
Cat.No: T12480
Synonym: Floropipamide,McN-JR 3345,酰胺哌啶酮,R 3345
Target: Others, Dopamine Receptor, 5-HT Receptor
Pipamperone HCl
Cat.No: T28417
Synonym: fluoropipamide,floropipamide hydrochloride,carpiperone,floropipamide,R4050,Pipamperone
Target:
TargetMol Loading
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