Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T4297 |
Flibanserin
BIMT-17BS,氟立班丝氨,Girosa,BIMT-17 |
Dopamine Receptor; 5-HT Receptor | GPCR/G Protein; Neuroscience |
Flibanserin (Girosa) 一种具有口服活性的 5-HT1A 受体激动剂和 5-HT2A 受体拮抗剂,Ki 值分别为 1 和 49 nM。它与多巴胺 D4 受体结合,Ki 值在 4 到 24 nM 之间。它是一种血清素能抗抑郁药,用于治疗性欲减退症。 | |||
T11295 |
Flibanserin-d4
BIMT-17BS D4,BIMT-17 D4,Flibanserin D4 |
Others | Others |
Flibanserin, a compound identified as BIMT-17, acts as a complete agonist at the serotonin 5-HT1A receptor, with a binding affinity (Ki) of 1 nM, while functioning as an antagonist at the 5-HT2A receptor with a 49 nM affinity. Flibanserin D4 represents a deuterium-labeled version of Flibanserin. | |||
T62324 |
Flibanserin hydrochloride
|
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Flibanserin (BIMT-17; BIMT-17BS) hydrochloride 是一种口服具有活力的 5-羟色胺的 5-HT1A 受体激动剂 (Ki: 1 nM) 和 5-HT2A (Ki: 49 nM) 受体拮抗剂。Flibanserin hydrochloride 同时可以结合多巴胺 D4 受体 (Ki: 4-24 nM)。Flibanserin hydrochloride 具有抗抑郁和抗焦虑的效果,能够用于性欲减退 (HSDD) 的研究。 |