4
2
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T3496 |
Buprofezin
噻嗪酮,NNI 750,Applaud,Buprofezine |
Reactive Oxygen Species | Immunology/Inflammation; Metabolism; NF-κB |
Buprofezin (Applaud) 是一种杀虫剂,通过抑制几丁质合成起作用,在体外还可以剂量依赖性地增加活性氧的产生。 | |||
T2256 |
CNX-1351
1-[4-[[2-(1H-吲唑-4-基)-4-(4-吗啉基)噻吩并[3,2-D]嘧啶-6-基]甲基]-1-哌嗪基]-6-甲基-5-庚烯-1,4-二酮 |
PI3K | PI3K/Akt/mTOR signaling |
CNX1351 是有效的、选择性的 PI3Kα 抑制剂,其 IC50=6.8 nM。 | |||
T3583 |
Macozinone
PBTZ169 |
Antibacterial; DprE1 | Microbiology/Virology; Others |
Macozinone (PBTZ169) 是具有杀菌作用的苯并噻嗪酮,也有抗结核作用。它也是一种 DprE1有效抑制剂,可通过与活性位点 Cys387 残基形成共价键来抑制必需的黄素蛋白 DprE1。 | |||
T79288 |
Antitubercular agent-38
|
||
Antitubercula agent-38,一种具有效抗结核活性的口服苯并噻嗪酮(BTZ)衍生物,其特点为低心脏毒性和低细胞毒性。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TN2312 |
Xanthiazone
|
Others | Others |
Xanthiazone is a natural product | |||
TN2313 |
Xanthiside
|
Others | Others |
Xanthiside is a natural product |