Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7218 |
Endomorphin 2
内吗啡肽 2 |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Endomorphin 2 是一种高亲和力和选择性的 μ-阿片受体激动剂,对 kappa3 结合位点具有合理的亲和力 ,Ki 为 20 到 30 nM 之间。 | |||
T11198 |
Endomorphin 2 TFA
|
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. a high affinity, highly selective agonist of the μ-opioid receptor, | |||
T73676 |
MIF-1 TFA
|
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MIF-1 TFA(Melanostatin)是一种内源性脑肽,具有有效调节多巴胺受体变构的作用,并抑制黑色素生成。此外,它通过阻断阿片受体的激活,调控吗啡的镇痛效果及应激诱导的镇痛(SIA)。MIF-1 TFA 能直接穿过血脑屏障(BBB)进入中枢神经系统。 |