Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
TP2077 |
α-Bungarotoxin
|
||
Neurotoxin that blocks neuromuscular transmission via irreversible inhibition of nicotinic ACh receptors (nAChRs). Prevents opening of nicotinic receptor-associated ion channels and is selective for α7 receptors over α3β4 receptors (IC50 values are 1.6 nM | |||
T80033 |
Biotin-α-Bungarotoxin
|
||
Biotin-α-Bungarotoxin是一种经Biotin标记的α-Bungarotoxin,后者是针对烟碱乙酰胆碱受体(nAChRs)的竞争性拮抗剂。 | |||
T80032 |
FITC-α-Bungarotoxin
|
||
FITC-α-Bungarotoxin为FITC标记之α-Bungarotoxin,该化合物为烟碱乙酰胆碱受体(nAChRs)竞争性拮抗剂。 | |||
T80466 |
κ-Bungarotoxin
κ-Bgt |
||
κ-Bungarotoxin (κ-Bgt) 是高效、特异性且缓慢可逆性α3β2神经元烟碱型乙酰胆碱受体(nAChR)拮抗剂,其IC50值为 2.30 nM。 | |||
T80167 |
αC-Conotoxin PrXA
αC-PrXA |
||
αC-Conotoxin PrXA为麻痹肽类神经毒素,亦是竞争性nAChR拮抗剂,对α1β1εδ(成人型)和α1β1γδ(胎儿型)nAChR的IC50值分别为1.8 nM和3.0 nM。该化合物通过与α-bungarotoxin竞争nAChR的α/δ及α/γ亚基界面,展现出对神经肌肉型nAChR的高度特异性。 |