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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T78878 |
α-Amylase/α-Glucosidase-IN-5
|
Glucosidase | Metabolism |
α-Amylase/α-Glucosidase-IN-5 (compound 4l) 是一种同时针对α-葡萄糖苷酶 (Glucosidase) 和α-淀粉酶 (Amylases) 的抑制剂,IC50 值分别为 5.96 μM 和 1.62 μM,显示出潜在的抗糖尿病活性。 | |||
T61706 |
α-Amylase/α-Glucosidase-IN-2
|
||
α-Amylase/α-Glucosidase-IN-2 (compound 5) exhibits strong inhibition activity towards both α-amylase and α-glucosidase enzymes, with IC 50 values of 13.02 μM and 13.09 μM, respectively. This compound shows promise for investigating diabetic complications [1]. | |||
T79402 |
α-Amylase/α-Glucosidase-IN-4
|
Glucosidase | Metabolism |
α-Amylase/α-Glucosidase-IN-4 (compound 5) 是一种针对 α-葡萄糖苷酶 (Glucosidase) 及 α-淀粉酶 (Amylases) 的双效抑制剂,分别展现出 0.15 μM 和 1.10 μM 的IC50s。该化合物展示了其潜在的抗糖尿病活性。 |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5690 |
7,4'-Di-O-methylapigenin
芹菜素二甲醚,4',7-DIMETHOXY-5-HYDROXYFLAVONE |
Amylase | Metabolism |
7,4'-Di-O-methylapigenin (4',7-DIMETHOXY-5-HYDROXYFLAVONE) 可能具有抗真菌c.zeyheri 的作用,是一种潜在的抗真菌药物。它还能抑制药物流出泵(IC50 = 51.64μg /毫升)。 |