Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T7173 |
[Leu5]-Enkephalin
亮氨酸脑啡肽,Leucine enkephalin,Leucyl-enkephalin,Leu-enkephalin |
Opioid Receptor; Endogenous Metabolite | Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience |
[Leu5]-Enkephalin (Leu-enkephalin) 是一种参与伤害感受的内源性神经肽,是 δ-阿片和 μ-阿片受体的激动剂,Ki 值分别为 4.0 和 3.4 nM | |||
T7665 |
[Leu5]-Enkephalin TFA(58822-25-6(free bas))
Leu-enkephalin,Leucine enkephalin,Leucyl-enkephalin |
Opioid Receptor; Endogenous Metabolite | Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience |
[Leu5]-Enkephalin TFA(58822-25-6(free bas)) (Leucyl-enkephalin) 是最有效的 δ 受体。 | |||
T22752L |
(D-Ser2)-Leu-Enkephalin-Thr
|
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
(D-Ser2)-Leu-Enkephalin-Thr 是阿片受体的 delta 选择性药物,具有镇痛作用。 | |||
T7173L |
[Leu5]-Enkephalin acetate(58822-25-6 free base)
亮氨酸脑啡肽,Leucine enkephalin,Leu-enkephalin,Leucyl-enkephalin |
Opioid Receptor; Endogenous Metabolite | Endocrinology/Hormones; GPCR/G Protein; Metabolism; Neuroscience |
[Leu5]-Enkephalin acetate(58822-25-6 free base) 是一种参与伤害感受的内源性神经肽,是 δ-opioid 和 μ-opioid 受体的激动剂(Kis 分别为 4.0 和 3.4 nM) | |||
TP1113L |
[Leu5]-Enkephalin, amide acetate
[Leu5]-Enkephalin, amide acetate(60117-24-0 free base) |
Opioid Receptor | Endocrinology/Hormones; GPCR/G Protein; Neuroscience |
[Leu5]-Enkephalin, amide acetate 是一种 δ 阿片受体激动剂。 | |||
T27878 |
LY 164929
LY-164929,LY164929 |
||
LY 164929 is a highly selective ligand for the lower affinity [3H]D-Ala2-D-Leu-5-enkephalin binding site. |