Cat. No. | Product Name | Target | Signaling Pathways |
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T36638 |
[Des-His1,Glu9]-Glucagon amide TFA
[Des-His1,Glu9]-Glucagon amide TFA |
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[Des-His1,Glu9]-Glucagon amide TFA is a potent peptide antagonist targeting the glucagon receptor, featuring a pA2 value of 7.2. It holds potential utility in diabetes pathogenesis research[1]. | |||
TP2033 |
[Des-His1,Glu9]-Glucagon amide
des-His1-[Glu9]-Glucagon (1-29) amide |
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Glucagon receptor antagonist (pA2 = 7.2 for inhibition of glucagon-induced adenylyl cyclase activation in rat liver membranes); displays no agonist activity. Enhances glucose-stimulated pancreatic insulin release in vitro. Blocks added glucagon-induced hy |