ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T1725 | Y-27632 dihydrochloride | 129830-38-2 | 320.26 | 10mM | Apoptosis; ROCK |
T1870 | Y-27632 | 146986-50-7 | 247.34 | 10mM | Apoptosis; ROCK |
T1898 | RKI-1447 | 1342278-01-6 | 326.37 | 10mM | ROCK |
T1911 | Afuresertib | 1047644-62-1 | 427.32 | 10mM | Akt; PKC; ROCK |
T2011 | RKI1313 | 1342276-76-9 | 340.4 | 10mM | ROCK |
T2155 | Thiazovivin | 1226056-71-8 | 311.36 | 10mM | ROCK |
T2482 | AT13148 | 1056901-62-2 | 313.78 | 10mM | Akt; PKA; ROCK; S6 Kinase; SGK |
T2633 | GSK429286A | 864082-47-3 | 432.37 | 10mM | ROCK |
T3060 | Fasudil hydrochloride | 105628-07-7 | 327.83 | 10mM | Autophagy; Calcium Channel; HIV Protease; PKA; PKC; ROCK; Serine/threonin kinase |
T3513 | GSK180736A | 817194-38-0 | 365.13 | 10mM | GRK; PKA; ROCK |
T3518 | GSK269962A | 850664-21-0 | 570.61 | 10mM | ROCK; S6 Kinase |
T4095 | ZINC00881524 | 557782-81-7 | 380.46 | 10mM | ROCK |
T4276 | Hydroxyfasudil Hydrochloride | 155558-32-0 | 343.83 | 10mM | ROCK |
T6057 | URMC-099 | 1229582-33-5 | 421.54 | 10mM | Aurora Kinase; Autophagy; Bcr-Abl; c-Met/HGFR; CDK; DNA Alkylation; IGF-1R; LRRK2; MEK; MLK; ROCK; SGK; Src; Syk; Trk receptor; VEGFR |
T6867 | Belumosudil | 911417-87-3 | 452.51 | 10mM | ROCK |
T4488 | GSK-25 | 874119-56-9 | 513.34 | 10mM | mTOR; ROCK; S6 Kinase |
T7301 | BDP5290 | 1817698-21-7 | 371.82 | 10mM | ROCK |
T7391 | SAR407899 | 923359-38-0 | 244.29 | 10mM | Rho; ROCK |
T7764 | CCG-222740 | 1922098-69-8 | 444.86 | 10mM | Ras; Rho; ROCK |
T7885 | Afuresertib hydrochloride | 1047645-82-8 | 463.8 | 10mM | Akt; PKC; ROCK |
TQ0319 | Ripasudil | 887375-67-9 | 395.88 | 10mM | ROCK |
T13384L | Y-33075 dihydrochloride | 173897-44-4 | 353.25 | 10mM | CaMK; PKC; ROCK |
T12746 | ROCK inhibitor-2 | 1127308-52-4 | 332.4 | 10mM | ROCK |
T10358 | Netarsudil hydrochloride | 1253952-02-1 | 526.45 | 10mM | ROCK |
T4276L | Hydroxyfasudil | 105628-72-6 | 307.37 | 10mM | PKA; ROCK |
TQ0187 | SR-3677 | 1072959-67-1 | 408.45 | 10mM | Autophagy; ROCK |
TQ0110 | ROCK-IN-2 | 867017-68-3 | 402.79 | 10mM | ROCK |
T23308 | SAR407899 hydrochloride | 923262-96-8 | 280.75 | 10mM | ROCK |
T14960 | Chroman 1 | 1273579-40-0 | 436.5 | 10mM | ROCK |
T12747 | ROCK2-IN-2 | 1995065-79-6 | 360.39 | 10mM | ROCK |
T12721 | Rho-Kinase-IN-1 | 1035094-83-7 | 352.5 | 10mM | ROCK |