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P450 inhibitor kit

Catalog No. CL0066

P450 inhibitor kit 包含细胞色素 P450抑制剂,P450是含有血红素作为单加氧酶的辅助因子的酶,在哺乳动物中,这些酶氧化类固醇、脂肪酸和异生物质,对于各种化合物的清除以及激素的合成和分解均很重要。TargetMol 为您提供83种精选 P450抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。

TargetMol的所有产品和服务仅用于科学研究,不能被用于人体,我们也不向个人提供产品和服务。
P450 inhibitor kit
规格 价格/CNY 货期 数量
10 μL * 10 mM (in DMSO) ¥ 1,992 4-6周
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产品组成

IDCompoundCASMWConcentrationTarget
T0603Phthalic acid mono-2-ethylhexyl ester4376-20-9278.3410mMEndogenous Metabolite; P450
T0679Ketoconazole65277-42-1531.4310mMAntifungal; Hydroxylase; NADPH-oxidase; P450; Ras
T0765Fomepizole7554-65-682.110mMAChR; CAT; P450
T1274Benzbromarone3562-84-3424.0810mMApoptosis; P450; Xanthine Oxidase
T1434Clarithromycin81103-11-9747.9510mMAntibacterial; Antibiotic; Autophagy; MRP; P450; ribosome
T1561Clobetasol propionate25122-46-7466.9710mMGlucocorticoid Receptor; P450
T1597Proadifen hydrochloride62-68-0389.9610mMP450
T1704Diosmetin520-34-3300.2610mMP450; Trk receptor
T2175Apigenin520-36-5270.2410mMAutophagy; P450
T2753Avasimibe166518-60-1501.7210mMAcyltransferase; P450
T2761Naringin dihydrochalcone18916-17-1582.5510mMNF-κB; P450
T2770Gentiopicroside20831-76-9356.3310mMHCV Protease; P450
T2949Alizarin72-48-0240.2210mMP450
T3002Piperine94-62-2285.3510mMAutophagy; Endogenous Metabolite; P-gp; P450
T3149Salvianolic Acid C115841-09-3492.4310mMP450
T3401Ginsenoside F153963-43-2638.8810mMEndogenous Metabolite; P450
T3411Curdione13657-68-6236.3410mMP450
T3417Amentoflavone1617-53-4538.4610mMAntibacterial; Antifungal; Apoptosis; COX; Opioid Receptor; P450; Phospholipase; Reactive Oxygen Species; RSV
T3585TMS24144-92-1300.3510mMP450
T3668Galangin548-83-4270.210mMAutophagy; ERK; NF-κB; P450
T3669Curcumenol19431-84-6234.310mMP450
T3735Tetrahydrocurcumin36062-04-1372.4110mMAutophagy; Endogenous Metabolite; P450
T3736Olivetol500-66-3180.2410mMCannabinoid Receptor; IκB/IKK; P450
T3776Rhapontigenin500-65-2258.310mMAntibacterial; Antifungal; P450
T4188SDZ285428174262-13-6401.8910mMAntifungal; P450; Parasite
T6050TAK-700426219-18-3307.3510mMP450
T6215Abiraterone Acetate154229-18-2391.5510mMP450
T6216Abiraterone154229-19-3349.5110mMP450
T6246Cobicistat1004316-88-4776.0210mMHIV Protease; P450
T6509Galeterone851983-85-2388.5510mMAndrogen Receptor; P450
T2S0663Humantenmine82354-38-9326.3910mMP450
T2S1434Bergaptol486-60-2202.1610mMP450
T5S0669Bergamottin7380-40-7338.410mMP450
T5S2343Acetylshikonin24502-78-1330.3310mMAChE; P450
T5S2360Corydaline518-69-4369.4610mMAChE; Opioid Receptor; P450; Virus Protease
T6S1894Linderane13476-25-0260.2810mMP450
T4498Stiripentol49763-96-4234.2910mMP450
T4567Sulfaphenazole526-08-9314.3610mMAntibacterial; P450
T7056Dronedarone141626-36-0556.7610mMAChR; Adrenergic Receptor; Autophagy; Calcium Channel; P450; Potassium Channel; Sodium Channel
T7088Diflubenzuron35367-38-5310.6810mMP450
T4S0800Demethyleneberberine25459-91-0324.3510mMAMPK; HIF; NF-κB; NOS; P450
T5582β-​Apo-​8'-​carotenal1107-26-2416.6410mMP450
T5594Cedrol77-53-2222.3710mMAntifungal; P450
T59531-Aminobenzotriazole1614-12-6134.1410mMP450
T74271-Ethynylnaphthalene15727-65-8152.1910mMP450
T7370Talarozole201410-53-9377.5110mMAutophagy; P450; Retinoid Receptor
T7410Furafylline80288-49-9260.2510mMP450
T74727-Hydroxyflavone6665-86-7238.2410mMP450
T8125Quinidine sulfate dihydrate6591-63-5782.910mMP450
TN1023Miltirone27210-57-7282.3810mMGABA Receptor; P450
T8729DMU21051031063-36-1259.310mMP450
T8728DMU2139104890-70-2289.310mMP450
TQ0296LN-Nornuciferine hydrochloride(4846-19-9 free base)TQ0296L317.8110mMP450
TN1702Glycycoumarin94805-82-0368.3710mMAutophagy; JNK; P450
T10953Dafadine-A1065506-69-5391.4610mMP450
T8937Soticlestat1429505-03-2373.4610mMP450
T11847LLiarozole115575-11-6308.7610mMP450; Retinoid Receptor
T9043AS1810722909561-15-5477.5210mMP450; STAT
TN13438-Geranyloxypsoralen7437-55-0338.410mMAnti-infection; BACE; P450
T16412Oteseconazole1340593-59-0527.3910mMAntifungal; P450
T17022Tebuconazole107534-96-3307.8210mMAntifungal; P450
T11991Mefentrifluconazole1417782-03-6397.7810mMAntifungal; P450
T14983Clomethiazole533-45-9161.6510mMGABA Receptor; P450
T215077-Ethoxyresorufin5725-91-7241.2410mMNO Synthase; P450
T21482Uniconazole83657-22-1291.7810mMP450; ROS Kinase
T9328Ellagic Acid Dihydrate133039-73-3338.2210mMP450
T50053Lofemizole65571-68-8192.6510mMP450
T220032,3-dihydrothieno-Thiadiazole Carboxylate152467-47-5200.2410mMP450
T14841BVT94839674-97-0241.2410mMHistone Methyltransferase; P450; phosphatase
T11680Isoasatone A67451-73-4448.5110mMP450
T21425Mephenytoin50-12-4218.2510mMP450
TN6848Piperonylic acid94-53-1166.1310mMP450
T97041-Ethynylpyrene34993-56-1226.2710mMP450
T22391Omeprazole Sodium95510-70-6368.4110mMProton pump;Autophagy;Antibacterial;P450
T377842,6-Dimethylquinoline877-43-0157.2110mMP450
T37826CAY10462502656-68-0360.3210mMP450
T10632Bucolome841-73-6266.3410mMP450;Immunology/Inflammation related
T10922CYP11B2-IN-11356479-78-1311.3510mMP450
T10335Antihistamine-11186430-60-3389.4710mMP450
T41291MS-PPOH206052-02-0323.4110mMP450
T10923CYP17-IN-12093317-51-0312.410mMP450
T15641K777233277-99-1574.7310mMCysteine Protease;P450;CCR
T21548PF-49815171390637-82-7456.5910mMP450

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包装与运输

  • DMSO溶液置于96孔板中
  • 蓝冰或干冰运输
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