PKA/cAMP inhibitor/activator kit 包含 PKA/cAMP 抑制剂/激活剂,G 蛋白偶联受体首先将信号传至腺苷酸环化酶,调节 cAMP 的含量,cAMP 决定PKA 的活性,PKA 负责很多蛋白的磷酸化,比如受体、离子通道、转录因子等,这是细胞快速应答胞外信号的过程。还有一类细胞缓慢应答胞外信号的过程,是cAMP 信号通路对细胞基因表达的影响。TargetMol 为您提供34种精选PKA/cAMP 抑制剂/激活剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0465 | Ellagic acid | 476-66-4 | 302.19 | 10mM | Carbonic Anhydrase; Casein Kinase; Endogenous Metabolite; Hedgehog/Smoothened; PKA; PKC; Reactive Oxygen Species; Syk; Topoisomerase |
T0610 | Piceatannol | 10083-24-6 | 244.24 | 10mM | Apoptosis; Autophagy; PKA; PKC; Serine/threonin kinase; Syk |
T0830 | Bithionol | 97-18-7 | 356.04 | 10mM | cAMP; Parasite |
T1418 | Bucladesine sodium | 16980-89-5 | 491.37 | 10mM | PDE; PKA |
T1920 | Capivasertib | 1143532-39-1 | 428.92 | 10mM | Akt; Autophagy; mTOR; PKA |
T2205 | Acefylline | 652-37-9 | 238.2 | 10mM | Adenosine Receptor; HDAC; PAD; PDE; PKA; TNF |
T2244 | ESI-09 | 263707-16-0 | 330.77 | 10mM | cAMP; Virus Protease |
T2356 | Ro-3306 | 872573-93-8 | 351.45 | 10mM | Apoptosis; CDK; ERK; PKA; PKC; SGK |
T2482 | AT13148 | 1056901-62-2 | 313.78 | 10mM | Akt; PKA; ROCK; S6 Kinase; SGK |
T2851 | Daphnetin | 486-35-1 | 178.14 | 10mM | Autophagy; EGFR; Parasite; PKA; PKC |
T3050 | ML-7 hydrochloride | 110448-33-4 | 452.74 | 10mM | Myosin; PKA; PKC; Serine/threonin kinase; YAP |
T3060 | Fasudil hydrochloride | 105628-07-7 | 327.83 | 10mM | Autophagy; Calcium Channel; HIV Protease; PKA; PKC; ROCK; Serine/threonin kinase |
T3269 | Metadoxine | 74536-44-0 | 298.29 | 10mM | 5-HT Receptor; PKA |
T4444 | A-674563 HCl (552325-73-2(free base)) | T4444 | 394.9 | 10mM | Akt; CDK; ERK; PKA; PKC |
T6250 | H-89 dihydrochloride | 130964-39-5 | 519.28 | 10mM | Autophagy; PKA; S6 Kinase |
T6304 | AT7867 | 857531-00-1 | 337.85 | 10mM | Akt; PKA; S6 Kinase |
T6536 | HJC0350 | 885434-70-8 | 277.38 | 10mM | cAMP |
T6680 | Staurosporine | 62996-74-1 | 466.53 | 10mM | Antibacterial; Antibiotic; Antifungal; Apoptosis; PKA; PKC; Src |
T6747 | 8-Bromo-cAMP sodium salt | 76939-46-3 | 430.08 | 10mM | PKA |
T4S2128 | Bilobetin | 521-32-4 | 552.49 | 10mM | PKA; PPAR |
T7648 | HA-100 | 84468-24-6 | 277.34 | 10mM | Myosin; PKA; PKC |
T15485 | HJC0197 | 1383539-73-8 | 339.45 | 10mM | cAMP; Ras |
T14069 | A-3 hydrochloride | 78957-85-4 | 321.22 | 10mM | CaMK; Casein Kinase; PKA; PKC |
TN1334 | 7-Methoxyrosmanol | 113085-62-4 | 360.45 | 10mM | cAMP |
T6139L | A-674563 2HCl(552325-73-2(fb-2hcl)) | T6139L | 431.36 | 10mM | Akt; CDK; ERK; PKA; PKC |
T15247 | ESI-05 | 5184-64-5 | 274.38 | 10mM | cAMP |
TP1789L | Malantide acetate(86555-35-3 free base) | TP1789L | 1693.97 | 10mM | PKA; PKC |
T12616L | CE3F4 | 143703-25-7 | 351.01 | 10mM | cAMP |
T15658 | KH7 | 330676-02-3 | 419.3 | 10mM | AChR; cAMP |
T21983L | PKI 14-22 amide, myristoylated Acetate | T21983L | 1269.54 | 10mM | PKA |
T21674L | PKA inhibitor fragment (6-22) amide Acetate | T21674L | 1928.11 | 10mM | PKA |
T9613 | TDI-10229 | T9613 | 313.79 | 10mM | cAMP |
T27525 | HA-1004 | 91742-10-8 | 293.35 | 10mM | PKA;PKC;Serine/threonin kinase |
T11212 | EPAC 5376753 | 302826-61-5 | 367.21 | 10mM | cAMP |