HER2 inhibitor kit 包含人表皮生长因子受体HER 抑制剂,HER2在正常细胞中的表达水平非常低,但是在胚胎发育期表达量非常高,对细胞发育过程的增殖、分化、迁移等起重要的作用,HER2的过量表达和许多上皮细胞癌症的恶化程度密切相关。TargetMol 为您提供28种精选HER2抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T1773 | Afatinib Dimaleate | 850140-73-7 | 718.08 | 10mM | Autophagy; EGFR; HER |
T2303 | Afatinib | 439081-18-2 | 485.94 | 10mM | EGFR; HER |
T2364 | Tucatinib | 937263-43-9 | 480.52 | 10mM | EGFR; HER |
T2630 | Poziotinib | 1092364-38-9 | 491.34 | 10mM | Apoptosis; EGFR; HER |
T3108 | CUDC-101 | 1012054-59-9 | 434.49 | 10mM | EGFR; HDAC; HER |
T3673 | Mollugin | 55481-88-4 | 284.3 | 10mM | HER; JAK |
T4342 | PF-04929113 Mesylate | 1173111-67-5 | 617.63 | 10mM | HER; HSP |
T6341 | PF04929113 | 908115-27-5 | 521.53 | 10mM | HER; HSP |
T6712 | Tyrphostin AG 879 | 148741-30-4 | 316.46 | 10mM | Apoptosis; EGFR; HER; PDGFR; Trk receptor |
T4S0544 | Furanodienone | 24268-41-5 | 230.3 | 10mM | Apoptosis; HER |
T7819 | TAS0728 | 2088323-16-2 | 504.58 | 10mM | EGFR; HER |
T22431 | SU5204 | 186611-11-0 | 265.31 | 10mM | EGFR; HER; VEGFR |
T11213 | Epertinib hydrochloride | 2071195-74-7 | 596.48 | 10mM | EGFR; HER |
T9072 | Tuxobertinib | 2414572-47-5 | 561.03 | 10mM | BTK; EGFR; HER; RIP kinase |
T9304 | (S)-Sunvozertinib | 2370013-49-1 | 584.09 | 10mM | EGFR; HER |
T34760 | SYR127063 | 871026-18-5 | 492.88 | 10mM | EGFR; HER |
T12594 | Pyrotinib dimaleate | 1397922-61-0 | 815.22 | 10mM | EGFR; HER |
T13088 | Tarloxotinib bromide | 1636180-98-7 | 681.77 | 10mM | EGFR;HER |
T4014 | CP-724714 | 383432-38-0 | 469.54 | 10mM | Apoptosis; EGFR |
T6124 | Mubritinib | 366017-09-6 | 468.47 | 10mM | EGFR; FGFR; JAK; PDGFR |
T6719 | Varlitinib | 845272-21-1 | 466.94 | 10mM | EGFR |
T8151 | Mobocertinib | 1847461-43-1 | 585.71 | 10mM | EGFR |
T21312 | Afatinib | 850140-72-6 | 485.94 | 10mM | Autophagy; EGFR |
T8758 | Poziotinib hydrochloride | 1429757-68-5 | 527.8 | 10mM | EGFR |
T27307 | Fasnall | 929978-58-5 | 338.47 | 10mM | Fatty Acid Synthase |
T9996 | NCT-58 | 2411429-33-7 | 466.57 | 10mM | HSP |
T2116 | AEE788 | 497839-62-0 | 440.58 | 10mM | Apoptosis; Bcr-Abl; c-Fms; EGFR; FLT |
T2483 | Dacomitinib | 1110813-31-4 | 469.94 | 10mM | Apoptosis; EGFR |