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Bcr-Abl inhibitor/degrader kit

Catalog No. CL0120

Bcr-Abl inhibitor/degrader kit 包含Bcr-Abl 抑制剂/降解剂,Bcr-Abl 融合基因是一种抗细胞凋亡的基因,具有高度酪氨酸激酶活性,促进细胞过度增殖,使细胞调控紊乱。Bcr-Abl 抑制剂/降解剂常用于慢性粒细胞白血病和其他肿瘤或疾病的治疗研究。TargetMol 为您提供50种精选Bcr-Abl 抑制剂/降解剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。

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Bcr-Abl inhibitor/degrader kit
规格 价格/CNY 货期 数量
10 μL * 10 mM (in DMSO) ¥ 1,500 4-6周
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产品组成

IDCompoundCASMWConcentrationTarget
T0152Bosutinib380843-75-4530.4510mMAutophagy; Bcr-Abl; Src
T1448Dasatinib302962-49-8488.0110mMApoptosis; Autophagy; Bcr-Abl; c-Kit; Src
T1448LDasatinib monohydrate863127-77-9506.0310mMApoptosis; Autophagy; Bcr-Abl; c-Kit; Ephrin Receptor; Src
T1524Nilotinib641571-10-0529.5210mMAutophagy; Bcr-Abl
T1621Imatinib Mesylate220127-57-1589.7110mMAutophagy; Bcr-Abl; c-Kit; PDGFR
T1803GNF-5778277-15-9418.3710mMBcr-Abl; SARS-CoV
T1817GNF-2778270-11-4374.3210mMBcr-Abl; SARS-CoV
T2070Agerafenib1188910-76-0517.4610mMBcr-Abl; c-Kit; c-RET; PDGFR; Raf; Src
T2094Danusertib827318-97-8474.5510mMAurora Kinase; Autophagy; Bcr-Abl; c-RET; FGFR; Trk receptor
T2116AEE788497839-62-0440.5810mMApoptosis; Bcr-Abl; c-Fms; EGFR; FLT
T2328Radotinib926037-48-1530.510mMBcr-Abl
T2341KW-24491000669-72-6332.410mMApoptosis; Aurora Kinase; Bcr-Abl; c-Kit; FGFR; FLT; JAK; Src
T2372Ponatinib943319-70-8532.5610mMAutophagy; Bcr-Abl; c-Kit; FGFR; PDGFR; Src; VEGFR
T2415PP1211092788-83-4319.3610mMApoptosis; Bcr-Abl; Hck; mTOR; PDGFR; Src; VEGFR
T2429Olverembatinib dimesylate1421783-64-3724.7710mMBcr-Abl
T2609Masitinib790299-79-5498.6410mMApoptosis; Bcr-Abl; c-Fms; c-Kit; FAK; FGFR; Hck; PDGFR; Src
T2640Rebastinib1020172-07-9553.5910mMApoptosis; Bcr-Abl; FLT; Src
T2802Nocodazole31430-18-9301.3210mMApoptosis; Autophagy; Bcr-Abl; CRISPR/Cas9; Microtubule Associated
T2920Berbamine dihydrochloride6078-17-7681.6510mMApoptosis; Autophagy; Bcr-Abl; NF-κB
T3063PD173955260415-63-2443.3510mMApoptosis; Bcr-Abl; Src
T3068AT9283896466-04-9381.4310mMApoptosis; Aurora Kinase; Autophagy; Bcr-Abl; FLT; JAK
T3071Olverembatinib1257628-77-5532.5710mMBcr-Abl
T3196GNF-7839706-07-9547.5310mMAChR; ACK; Bcr-Abl
T3641NVP-BAW2881861875-60-7424.3810mMBcr-Abl; Raf; VEGFR
T4053AST 487630124-46-8529.5610mMBcr-Abl; c-Kit; c-RET; FLT; VEGFR
T4191Multi-kinase inhibitor 1778274-97-8418.3810mMBcr-Abl; c-Kit; PDGFR
T4320Flumatinib895519-90-1562.610mMBcr-Abl; c-Kit; PDGFR
T6196PP1172889-26-8281.3610mMApoptosis; Bcr-Abl; c-Kit; EGFR; Src
T6230Imatinib152459-95-5493.610mMAutophagy; Bcr-Abl; c-Kit; PDGFR; SARS-CoV
T6300Degrasyn856243-80-6384.2710mMApoptosis; Autophagy; Bcr-Abl; DUB
T6311Bafetinib859212-16-1576.6210mMAutophagy; Bcr-Abl; Src
T6348NVP-BHG712940310-85-0503.4910mMBcr-Abl; Ephrin Receptor; Raf; Src
T5177Asciminib1492952-76-7449.8410mMBcr-Abl
T7186CZC-8004916603-07-1309.3410mMBcr-Abl
T7861Flumatinib mesylate895519-91-2658.6910mMBcr-Abl; c-Kit; PDGFR
T8488GMB-4752490599-18-1861.9310mMBcr-Abl
T11916Lyn-IN-1887650-05-7576.610mMBcr-Abl; Src
T2147Nilotinib monohydrochloride monohydrate923288-90-8583.9910mMAutophagy; Bcr-Abl
T16750Rigosertib592542-59-1451.4910mMApoptosis; Bcr-Abl; CDK; FLT; PDGFR; PI3K; PLK; Src
T8882Vodobatinib1388803-90-4453.9210mMBcr-Abl
T17267XL228898280-07-4437.5410mMAurora Kinase; Bcr-Abl; IGF-1R; Src
T11641N-Desmethyl imatinib404844-02-6479.5810mMBcr-Abl; c-Kit; Drug Metabolite; PDGFR
T21785AG957140674-76-6273.2810mMBcr-Abl
T16545Pivanex122110-53-6202.2510mMApoptosis; Bcr-Abl; HDAC
T11960MBM-552083622-09-5498.5510mMMAPK;S6 Kinase;DYRK;Chk;GSK-3;Bcr-Abl;Akt;Aurora Kinase;CDK
T12310ON 1460401404231-34-0489.5510mMPI3K;Bcr-Abl
T30855CGP77675234772-64-6443.5410mMEGFR;VEGFR;Src;Bcr-Abl
T11961MBM-55S2083624-07-9734.7310mMMAPK;S6 Kinase;GSK-3;Bcr-Abl;CDK;CDK;Akt;Aurora Kinase
T10799CHMFL-ABL-0392304344-56-5594.6310mMBcr-Abl
T10800CHMFL-ABL-1212270879-07-5580.6710mMBcr-Abl

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产品应用

  • 信号通路研究
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包装与运输

  • DMSO溶液置于96孔板中
  • 蓝冰或干冰运输
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