Powder: -20°C for 3 years | In solvent: -80°C for 1 year
Otamixaban(FXV673) is an effective (Ki = 0.5 nM), selective, rapid-acting, competitive, and reversible fXa inhibitor. It also effectively inhibits both free and prothrombinase-bound fXa.
规格 | 价格/CNY | 货期 | 数量 | |
---|---|---|---|---|
2 mg | ¥ 1,290 | 5日内发货 | ||
5 mg | ¥ 2,230 | 5日内发货 | ||
25 mg | ¥ 7,690 | 6-8周 | ||
50 mg | ¥ 9,990 | 6-8周 | ||
100 mg | ¥ 15,500 | 6-8周 |
产品描述 | Otamixaban(FXV673) is an effective (Ki = 0.5 nM), selective, rapid-acting, competitive, and reversible fXa inhibitor. It also effectively inhibits both free and prothrombinase-bound fXa. |
体内活性 | Otamixaban is highly efficacious in rodent, canine and porcine models of thrombosis showed in vivo experiments. Recent clinical findings indicate that Otamixaban is efficacious, safe, and well-tolerated in humans and therefore has considerable potential for the treatment of acute coronary syndrome. |
别名 | FXV673, 奥米沙班 |
分子量 | 446.5 |
分子式 | C25H26N4O4 |
CAS No. | 193153-04-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 50 mg/mL (111.98 mM), Sonication is recommended.
可选溶剂 | 浓度 体积 质量 | 1 mg | 5 mg | 10 mg | 25 mg |
DMSO | 1 mM | 2.2396 mL | 11.1982 mL | 22.3964 mL | 55.991 mL |
5 mM | 0.4479 mL | 2.2396 mL | 4.4793 mL | 11.1982 mL | |
10 mM | 0.224 mL | 1.1198 mL | 2.2396 mL | 5.5991 mL | |
20 mM | 0.112 mL | 0.5599 mL | 1.1198 mL | 2.7996 mL | |
50 mM | 0.0448 mL | 0.224 mL | 0.4479 mL | 1.1198 mL | |
100 mM | 0.0224 mL | 0.112 mL | 0.224 mL | 0.5599 mL |
对于不同动物的给药剂量换算,您也可以参考 更多...
请在以下方框中输入您的动物实验信息后点击计算,可以得到母液配置方法和体内配方的制备方法: 比如您的给药剂量是10 mg/kg,每只动物体重20 g,给药体积100 μL,一共给药动物10 只,您使用的配方为5% DMSO+30% PEG300+5% Tween 80+60% ddH2O。那么您的工作液浓度为2 mg/mL。
母液配置方法:2 mg 药物溶于 50 μL DMSO (母液浓度为 40 mg/mL), 如您需要配置的浓度超过该产品的溶解度,请先与我们联系。
体内配方的制备方法:取 50 μL DMSO 主液,加入 300 μL PEG300, 混匀澄清,再加 50 μL Tween 80,混匀澄清,再加 600 μL ddH2O, 混匀澄清。
您可能有的问题的答案可以在抑制剂处理说明中找到,包括如何准备库存溶液,如何存储产品,以及基于细胞的分析和动物实验需要特别注意的问题。
Otamixaban 193153-04-7 Others FXV 673 FXV-673 FXV673 奥米沙班 Inhibitor inhibitor inhibit