Powder: -20°C for 3 years | In solvent: -80°C for 1 year
GPR40 agonist 4 is a potent free fatty acid agonist of receptor 1 (pEC50: 7.54).
规格 | 价格/CNY | 货期 | 数量 | |
---|---|---|---|---|
2 mg | ¥ 591 | 5日内发货 | ||
5 mg | ¥ 997 | 6-8周 | ||
10 mg | ¥ 1,490 | 6-8周 | ||
25 mg | ¥ 3,440 | 6-8周 | ||
100 mg | ¥ 6,240 | 6-8周 | ||
1 mL * 10 mM (in DMSO) | ¥ 913 | 6-8周 |
产品描述 | GPR40 agonist 4 is a potent free fatty acid agonist of receptor 1 (pEC50: 7.54). |
靶点活性 | FFA1/GPR40:(pEC50)7.54 |
体外活性 | GPR40 agonist 4 has a low risk of activating caspase-3/7. |
体内活性 | The area under the curve of blood glucose (AUC0-120min) and blood insulin (AUC0-120min) reveal that the minimum effective dose of GPR40 agonist 4 is 3 mg/kg. The hyperglycemia state is also markedly improved in GPR40 agonist 4 (20 mg/kg) treated group. When GPR40 agonist 4 is dosed 60 min prior to the oral glucose challenge, single oral administration of GPR40 agonist 4 robustly decreases the plasma glucose excursion and enhances insulin secretion during an oral glucose tolerance test (OGTT) in a dose-dependent manner from 1 to 10 mg/kg. |
分子量 | 416.87 |
分子式 | C21H17ClO5S |
CAS No. | 2102196-57-4 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
DMSO: 160 mg/mL (383.81 mM), Sonication and heating are recommended.
可选溶剂 | 浓度 体积 质量 | 1 mg | 5 mg | 10 mg | 25 mg |
DMSO | 1 mM | 2.3988 mL | 11.9941 mL | 23.9883 mL | 59.9707 mL |
5 mM | 0.4798 mL | 2.3988 mL | 4.7977 mL | 11.9941 mL | |
10 mM | 0.2399 mL | 1.1994 mL | 2.3988 mL | 5.9971 mL | |
20 mM | 0.1199 mL | 0.5997 mL | 1.1994 mL | 2.9985 mL | |
50 mM | 0.048 mL | 0.2399 mL | 0.4798 mL | 1.1994 mL | |
100 mM | 0.024 mL | 0.1199 mL | 0.2399 mL | 0.5997 mL |
对于不同动物的给药剂量换算,您也可以参考 更多...
请在以下方框中输入您的动物实验信息后点击计算,可以得到母液配置方法和体内配方的制备方法: 比如您的给药剂量是10 mg/kg,每只动物体重20 g,给药体积100 μL,一共给药动物10 只,您使用的配方为5% DMSO+30% PEG300+5% Tween 80+60% ddH2O。那么您的工作液浓度为2 mg/mL。
母液配置方法:2 mg 药物溶于 50 μL DMSO (母液浓度为 40 mg/mL), 如您需要配置的浓度超过该产品的溶解度,请先与我们联系。
体内配方的制备方法:取 50 μL DMSO 主液,加入 300 μL PEG300, 混匀澄清,再加 50 μL Tween 80,混匀澄清,再加 600 μL ddH2O, 混匀澄清。
您可能有的问题的答案可以在抑制剂处理说明中找到,包括如何准备库存溶液,如何存储产品,以及基于细胞的分析和动物实验需要特别注意的问题。
GPR40 agonist 4 2102196-57-4 Others GPR-40 agonist 4 Inhibitor inhibitor inhibit