Ras inhibitor kit 包含Ras 抑制剂,Ras 蛋白是原癌基因c-Ras 的表达产物,属于GTPase 家族,参与了RAF-MEK-ERK 这条调节通路的传导,调控基因转录过程从而影响细胞增殖、调亡、分化和肿瘤细胞的生存、增值、迁移、扩散、血管生成等。TargetMol 为您提供34种精选Ras 抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T1876 | Kobe0065 | 436133-68-5 | 449.79 | 10mM | Apoptosis; Raf; Ras |
T6163 | Salirasib | 162520-00-5 | 358.54 | 10mM | Autophagy; Ras |
T6302 | Lonafarnib | 193275-84-2 | 638.82 | 10mM | Autophagy; Raf; Ras; Transferase |
T6462 | Deltarasin | 1440898-61-2 | 603.75 | 10mM | PDE; Ras |
T6555 | K-Ras(G12C) inhibitor 12 | 1469337-95-8 | 449.67 | 10mM | Apoptosis; Raf; Ras |
T5418 | BAY-293 | 2244904-70-7 | 448.58 | 10mM | Raf; Ras |
T5469 | K-Ras-IN-1 | 84783-01-7 | 207.29 | 10mM | Raf; Ras |
T7131 | Antineoplaston A10 | 91531-30-5 | 246.26 | 10mM | Apoptosis; Endogenous Metabolite; Ras |
T7326 | 6H05 (TFA) | 2061344-88-3 | 590.14 | 10mM | Ras |
T7414 | ARS-853 | 1629268-00-3 | 432.94 | 10mM | Apoptosis; Raf; Ras |
T7609 | ARS-1620 | 1698055-85-4 | 430.84 | 10mM | Ras |
T7558 | CID-1067700 | 314042-01-8 | 390.48 | 10mM | Ras |
T8006 | Oncrasin-1 | 75629-57-1 | 269.73 | 10mM | Apoptosis; Raf; Ras |
T8369 | Adagrasib | 2326521-71-3 | 604.12 | 10mM | Ras |
T12979 | BI-3406 | 2230836-55-0 | 462.46 | 10mM | MAPK; p38 MAPK; Ras |
T8684 | Sotorasib | 2296729-00-3 | 560.59 | 10mM | Ras |
T16143 | MRTX-1257 | 2206736-04-9 | 565.71 | 10mM | Ras |
T8756 | KRAS inhibitor-9 | 300809-71-6 | 292.8 | 10mM | Apoptosis; Ras |
T8843 | APS6-45 | 2188236-41-9 | 548.4 | 10mM | MAPK; Ras |
T8870 | 1-(4-methansulfinylphenyl)ethanone | 32361-73-2 | 182.24 | 10mM | Ras |
T16021 | MBQ-167 | 2097938-73-1 | 338.41 | 10mM | CDK; Ras |
T9184L | Compound 3344 hydrochloride | T9184L | 426.94 | 10mM | Ras |
T9407 | Rasarfin | 674359-73-0 | 425.91 | 10mM | Ras |
T10376 | ARS-1630 | 1698055-86-5 | 430.83 | 10mM | Ras |
T11738 | K-Ras G12C-IN-4 | 2376328-55-9 | 561.07 | 10mM | Ras |
T16432 | Pan-RAS-IN-1 | 1835283-94-7 | 717.65 | 10mM | MAPK; Ras |
T20759 | XRP44X | 729605-21-4 | 380.87 | 10mM | Ras |
T10375 | ARS-1323 | 1698024-73-5 | 430.83 | 10mM | Ras |
T24437 | MCP110 | 521310-51-0 | 508.65 | 10mM | Ras;Raf |
T40186 | Garsorasib | 2559761-14-5 | 598.65 | 10mM | Ras |
T3725 | K-Ras(G12C) Inhibitor 6 | 2060530-16-5 | 405.33 | 10mM | Raf |
T3857 | magnolin | 31008-18-1 | 416.47 | 10mM | ERK |
T6556 | K-Ras(G12C) inhibitor 9 | 1469337-91-4 | 513.78 | 10mM | Raf |
T6948 | Pluripotin | 839707-37-8 | 550.53 | 10mM | ERK; Raf; S6 Kinase |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |