PDE inhibitor kit 包含磷酸二酯酶 PDE 抑制剂,PDE 抑制剂通过抑制 cAMP 的裂解,升高细胞内 cAMP 的浓度,增加钙离子内流,从而产生正性肌力的作用。另外,PDE 抑制剂通过增高血管平滑肌细胞内 cAMP 的含量起到扩血管的作用。TargetMol 为您提供86种精选 PDE 抑制剂。所有化合物现货供应,到货快捷,是您预实验探索的不二选择。
ID | Compound | CAS | MW | Concentration | Target |
---|---|---|---|---|---|
T0070 | Pentoxifylline | 6493-05-6 | 278.31 | 10mM | Adenosine Receptor; Autophagy; HIV Protease; PDE |
T0462 | Cilostazol | 73963-72-1 | 369.46 | 10mM | Autophagy; PDE |
T0467 | Sildenafil citrate | 171599-83-0 | 666.7 | 10mM | Apoptosis; Autophagy; PDE |
T1024 | Roflumilast | 162401-32-3 | 403.21 | 10mM | PDE; RSV |
T1027 | Luteolin | 491-70-3 | 286.24 | 10mM | Apoptosis; Autophagy; Endogenous Metabolite; PDE; Nrf2 |
T1096 | Milrinone | 78415-72-2 | 211.22 | 10mM | PDE |
T1265 | Amrinone | 60719-84-8 | 187.2 | 10mM | PDE; TNF |
T1398 | Tadalafil | 171596-29-5 | 389.4 | 10mM | Apoptosis; PDE |
T1681 | Aminophylline | 317-34-0 | 420.43 | 10mM | Adenosine Receptor; PDE |
T1708 | Pimobendan | 74150-27-9 | 334.37 | 10mM | PDE |
T1713 | IBMX | 28822-58-4 | 222.24 | 10mM | PDE |
T1745 | Balipodect | 1238697-26-1 | 428.42 | 10mM | PDE |
T2129 | Zaprinast | 37762-06-4 | 271.27 | 10mM | PDE |
T2137 | Ibudilast | 50847-11-5 | 230.51 | 10mM | PDE |
T2334 | Avanafil | 330784-47-9 | 483.95 | 10mM | PDE |
T2923 | Apremilast | 608141-41-9 | 460.5 | 10mM | Apoptosis; PDE; TNF |
T3987 | Lotamilast | 947620-48-6 | 472.17 | 10mM | PDE |
T4097 | Vardenafil hydrochloride trihydrate | 330808-88-3 | 579.11 | 10mM | PDE |
T4285 | Crisaborole | 906673-24-3 | 251.05 | 10mM | PDE |
T4462 | Roflumilast N-oxide | 292135-78-5 | 419.21 | 10mM | PDE |
T6042 | [11C]MP 10 | 1292799-56-4 | 392.45 | 10mM | PDE |
T6054 | GSK256066 | 801312-28-7 | 518.58 | 10mM | PDE |
T6445 | Cilomilast | 153259-65-5 | 343.42 | 10mM | PDE |
T6462 | Deltarasin | 1440898-61-2 | 603.75 | 10mM | PDE; Ras |
T6644 | Rolipram | 61413-54-5 | 275.34 | 10mM | Antibacterial; HIV Protease; PDE |
T6649 | (S)-(+)-Rolipram | 85416-73-5 | 275.34 | 10mM | Apoptosis; PDE |
T4695 | CP671305 | 445295-04-5 | 454.4 | 10mM | PDE |
T5033 | Olprinone | 106730-54-5 | 250.26 | 10mM | PDE |
T5106 | BRL-50481 | 433695-36-4 | 244.27 | 10mM | PDE |
T5101 | BW-A 78U | 101155-02-6 | 257.27 | 10mM | PDE |
T5474 | D159687 | 1155877-97-6 | 366.85 | 10mM | PDE |
T5956 | VP3.15 dihydrobromide | 1281681-33-1 | 528.3 | 10mM | GSK-3; PDE |
T6147 | Nortadalafil | 171596-36-4 | 375.38 | 10mM | PDE |
T5940 | Proxyphylline | 603-00-9 | 238.24 | 10mM | Adenosine Receptor; PDE |
T7346 | Lodenafil | 139755-85-4 | 504.6 | 10mM | PDE |
T7542 | Amino Tadalafil | 385769-84-6 | 390.39 | 10mM | PDE |
T7642 | Cilostamide | 68550-75-4 | 342.43 | 10mM | PDE |
T7954 | YM976 | 191219-80-4 | 313.78 | 10mM | PDE |
T5S2059 | Glaucine | 475-81-0 | 355.4 | 10mM | Adrenergic Receptor; Calcium Channel; Dopamine Receptor; Influenza Virus; PDE |
T8515 | Osoresnontrine | 1189767-28-9 | 311.34 | 10mM | PDE |
T8454 | SEP-0372814 | 1516895-53-6 | 369.42 | 10mM | PDE |
T8462 | Enoximone | 77671-31-9 | 248.3 | 10mM | PDE |
T8506 | THPP-1 | 1257051-63-0 | 464.9 | 10mM | PDE |
T5496 | ML-030 | 1013750-77-0 | 412.46 | 10mM | PDE |
T8659 | K-Ras-PDEδ-IN-1 | 1841464-21-8 | 447.5 | 10mM | PDE |
T16079 | Mirodenafil | 862189-95-5 | 531.67 | 10mM | PDE |
T17199 | Udenafil | 268203-93-6 | 516.66 | 10mM | PDE |
T8787 | Drotaverine hydrochloride | 985-12-6 | 433.97 | 10mM | PDE |
T21965 | MBCQ | 150450-53-6 | 313.74 | 10mM | PDE |
T8919 | Homo Sildenafil | 642928-07-2 | 488.6 | 10mM | PDE |
TN2159 | Robustine | 2255-50-7 | 215.2 | 10mM | PDE |
T10590 | Zatolmilast | 1606974-33-7 | 405.8 | 10mM | PDE |
T11689 | ITI-214 | 1642303-38-5 | 605.56 | 10mM | PDE |
T23256 | RS-25344 hydrochloride | 152815-28-6 | 411.8 | 10mM | PDE |
T9239 | RS-25344 | 152814-89-6 | 375.34 | 10mM | PDE |
T50062 | 2,5-dichloro-4-(difluoromethoxy)-N,N-dimethylbenzene-1-sulfonamide | 473477-26-8 | 320.14 | 10mM | PDE |
T12150 | N-Methylbenzamide | 613-93-4 | 135.16 | 10mM | PDE |
T12267 | NSP-805 | 125068-54-4 | 297.35 | 10mM | PDE |
T16499 | Mardepodect | 898562-94-2 | 392.45 | 10mM | PDE |
T16164 | MY-5445 | 78351-75-4 | 331.8 | 10mM | PDE |
T22851 | ICI 63197 | 27277-00-5 | 207.23 | 10mM | PDE |
T24656 | PQ-10 | 927691-21-2 | 403.43 | 10mM | PDE |
T19706 | Ro 20-1724 | 29925-17-5 | 278.35 | 10mM | PDE |
T19865 | GEBR-7b | 67387-76-2 | 220.26 | 10mM | PDE |
T23154 | Piclamilast | 144035-83-6 | 381.25 | 10mM | PDE |
T25376 | Ensifentrine | 1884461-72-6 | 477.56 | 10mM | PDE |
T27172 | Difamilast | 937782-05-3 | 446.44 | 10mM | PDE |
TN1416 | Ayanin | 572-32-7 | 344.32 | 10mM | P450;PARP;IL Receptor;PDE |
T12913 | Siguazodan | 115344-47-3 | 284.32 | 10mM | PDE |
T27475 | GSK356278 | 720704-34-7 | 439.53 | 10mM | PDE |
T9816 | Arofylline | 136145-07-8 | 304.73 | 10mM | PDE |
T21865 | BC 11-38 | 686770-80-9 | 304.43 | 10mM | PDE |
T28352 | PDE9-IN-(S)-C33 | 2066488-39-7 | 357.84 | 10mM | PDE |
T21457 | Carbazeran | 70724-25-3 | 360.41 | 10mM | PDE |
T13189 | TP-10 | 898563-00-3 | 460.45 | 10mM | PDE |
T9805 | BAY 2666605 | 2275774-60-0 | 352.28 | 10mM | PDE |
T15381 | Gisadenafil | 334826-98-1 | 519.62 | 10mM | PDE |
T39341 | FCPR03 | 1917347-65-9 | 299.31 | 10mM | PDE |
TN4510 | (+)-Medioresinol Di-O-β-D-glucopyranoside | 88142-63-6 | 712.69 | 10mM | PDE |
T9871 | Dazonone | 105622-85-3 | 235.67 | 10mM | PDE |
T11220L | UK 227786 | 150452-21-4 | 477.34 | 10mM | PDE |
T23638 | Adibendan | 100510-33-6 | 278.31 | 10mM | PDE |
T10730 | CDC801 | 192819-27-5 | 408.45 | 10mM | PDE;TNF |
T10841 | CM-675 | 1872466-47-1 | 536.62 | 10mM | PDE |
T14217 | AMG 579 | 1227067-61-9 | 441.48 | 10mM | PDE |
T12395 | PDE9-IN-1 | 2305087-92-5 | 362.4 | 10mM | PDE |
Empty | 1000025-07-9 | 1000413-72-8 | 229005-80-5 | 1000787-75-6 | 946387-07-1 | 1000998-59-3 | 1175526-27-8 | 1001288-58-9 | 1001350-96-4 | 1001404-83-6 | Empty |
Vadadustat | TAK875 | TAK-779 | Tegobuvir | RN-1734 | BMS-687453 | AM211 | FT011 | BMS754807 | AAI101 | ||
Empty | 1001625-82-6 | 1001645-58-4 | 1001753-24-7 | 1001908-89-9 | 1002304-34-8 | 1002-84-2 | 100291-86-9 | 100299-08-9 | 10030-52-1 | 10040-45-6 | Empty |
RPW-24 | SRT1720 hydrochloride | INH6 | SRT 2183 | AMG208 | Pentadecanoic acid | Apiopaeonoside | Pemirolast potassium | L-Anserine nitrate salt | Sodium Picosulfate | ||
Empty | 100427-26-7 | 1004316-88-4 | 10045-45-1 | 100462-37-1 | 1004990-28-6 | 100-51-6 | 1005-24-9 | 1005264-47-0 | 1005334-57-5 | 1005342-46-0 | Empty |
Lercanidipine | Cobicistat | 1-Ethyl-2-benzimidazolinone | ROSIRIDIN | PF-AKT400 | Benzyl alcohol | 1-Methylnicotinamide chloride | MX69 | CVT-10216 | LCL161 | ||
Empty | 1005491-05-3 | 100-55-0 | 1005504-62-0 | 1005883-72-6 | 100643-71-8 | 1007207-67-1 | 10075-50-0 | 1007647-73-5 | 100784-20-1 | 10083-24-6 | Empty |
Tirasemtiv | Roniacol | Rg3039 | Z433927330 | Desloratadine | CH5132799 | 5-Bromoindole | Smurf1-IN-A01 | Halosulfuron-methyl | Piceatannol | ||
Empty | 100872-83-1 | 100874-08-6 | 1009119-64-5 | 1009119-65-6 | 100929-71-3 | 1009298-09-2 | 1009298-59-2 | 100929-99-5 | 1009734-33-1 | 10097-84-4 | Empty |
ML346 | SB 4 | Daclatasvir | Daclatasvir dihydrochloride | NADPH (tetracyclohexanamine) | AZD8055 | Vistusertib | PAβN dihydrochloride | HZ1157 | Rotundine | ||
Empty | 1009816-48-1 | 1009817-63-3 | 1009820-21-6 | 100986-85-4 | 101001-34-7 | 1010411-21-8 | 1010-60-2 | 1011244-68-0 | 1011301-27-1 | 1011529-10-4 | Empty |
Thiamet G | B-AP15 | Silmitasertib | Levofloxacin | Pamicogrel | GSK369796 Dihydrochloride | 2-Chloronaphthoquinone | TFAP | Tenovin3 | Azvudine | ||
Empty | 101152-94-7 | 101155-02-6 | 1011557-82-6 | 1011-74-1 | 101-20-2 | 1012054-59-9 | 101-21-3 | 101-26-8 | 101303-98-4 | 1013101-36-4 | Empty |
Milnacipran hydrochloride | BW-A78U | Tenovin-6 | DL-Normetanephrine hydrochloride | Triclocarban | CUDC101 | Chlorpropham | Mestinon | Zacopride hydrochloride | PF04691502 | ||
Empty | 101-31-5 | 1013-69-0 | 1013750-77-0 | 1013753-99-5 | 10138-52-0 | 1013920-15-4 | 1013937-63-7 | 1014691-61-2 | 101477-54-7 | 101494-95-5 | Empty |
L-Hyoscyamine | Noreugenin | ML-030 | BC-1382 | Gadolinium chloride | Vorolanib | VTP-27999 TFA | GSK0660 | Lomerizine hydrochloride | 8-CHLOROQUINAZOLIN-4(1H)-ONE |