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Cat. No. Product Name Target Signaling Pathways
T0827 Cefsulodin sodium

Cefsulodine sodium,Sulcephalosporin,头孢磺啶钠

Antibacterial; Antibiotic Microbiology/Virology
Cefsulodin sodium (Sulcephalosporin) 是β内酰胺抗生素,对缘脓杆菌和肠杆菌有活性。
T12231 NITD-349

Others; Antibacterial Microbiology/Virology; Others
NITD-349 是MmpL3的抑制剂,它对毒性结核分枝杆菌 H37Rv 显示出高效的抗分枝杆菌活性,MIC50 为 23 nM。
T61067 MurB-IN-1

MurB-IN-1 (compound 44) is a potent inhibitor of MurB, an essential enzyme involved in the synthesis of bacterial cell wall. With a binding affinity of K d 3.57 μM, MurB-IN-1 effectively hinders the activity of MurB, presenting a promising therapeutic option against P. aeruginosa, a highly virulent and opportunistic pathogen associated with severe infections and mortality [1].
T81360 PSMα3 TFA

PSMα3 TFA 作为一种肽类化合物,主要用于诱导生成耐受性的树突细胞(DC),以应用于DC疫苗接种。该化合物能对TLR2和TLR4诱导的DC成熟过程进行调节,抑制促炎和消炎细胞因子的产生,降低抗原摄取,并影响人单核细胞来源DC的渗透和调节能力。此外,PSMα3 TFA 是耐甲氧西林金黄色葡萄球菌(MRSA)中最有毒株释放的关键毒素之一。

化合物

Cefsulodin sodium
Cat.No: T0827
Synonym: Cefsulodine sodium,Sulcephalosporin,头孢磺啶钠
Target: Antibacterial, Antibiotic
NITD-349
Cat.No: T12231
Synonym:
Target: Others, Antibacterial
MurB-IN-1
Cat.No: T61067
Synonym:
Target:
PSMα3 TFA
Cat.No: T81360
Synonym:
Target:
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