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Cat. No. Product Name Target Signaling Pathways
T3221 Oct3/4-inducer-1

2-(4-(4-methoxybenzyloxy)phenyl)acetonitrile,2-(4-[(4-甲氧基苄基)氧基]苯基)乙腈

Others; OCT Membrane transporter/Ion channel; Others
Oct3/4-inducer-1 (2-(4-(4-methoxybenzyloxy)phenyl)acetonitrile) 是Oct3/4诱导剂,能够促进 Oct3/4 的表达和稳定,提高其在多种人体细胞中的转录活性。
T68110 Moxnidazole

Moxnidazole 是一种5-硝基咪唑,在微生物试验和果蝇中具有诱变性,诱导小鼠体细胞的遗传改变。
TP1057L Phe-Met-Arg-Phe Like Peptide acetate

Pqdpflrfamide acetate,Phe-Met-Arg-Phe Like Peptide acetate(98495-35-3 free base)

Others Others
Phe-Met-Arg-Phe Like Peptide acetate (Pqdpflrfamide acetate)(98495-35-3 free base) 是一种来自蜗牛 Helix aspersa 的内脏和躯体肌肉的 FMRF 样肽。 FMRF (Phe-Met-Arg-Phe) 是一种由 4 个氨基酸残基组成的神经肽肽。
T8768 MM-102 TFA

HMTase Inhibitor IX TFA

Histone Methyltransferase Chromatin/Epigenetic
MM-102 TFA (HMTase Inhibitor IX TFA) 是一种有效的 WDR5/MLL 相互作用抑制剂,在 WDR5 结合检测中,IC50为 2.4 nM,Ki 小于 1 nM。
T23271 RSC-133

Others Others
promotes the reprogramming of human somatic cells to pluripotent stem cells
T82520 Dynorphin (2-17) (porcine)

Dynorphin (2-17) (porcine),一种源自Prodynorphin的肽类化合物,具有缓解Morphine依赖性戒断症状的功能。
TP1057 Phe-Met-Arg-Phe Like Peptide, Snail Helix aspersa

Phe-Met-Arg-Phe Like Peptide

Phe-Met-Arg-Phe-like peptide, derived from the visceral and somatic muscles of the snail Helix aspersa, is a neuropeptide known as FMRF (Phe-Met-Arg-Phe). This peptide comprises four amino acid residues[1].
T78520 CYT296

Others Others
CYT296是一种靶向染色质去凝集的化合物,能增强定义因子(OSKM)介导诱导多能干细胞(iPSC)的生成,并通过诱导小鼠胚胎成纤维细胞(MEFs)染色质的开放状态来促进体细胞的重编程,适用于细胞替代治疗和药物筛选的研究领域。
T63606 Cav 3.2 inhibitor 2

Cav 3.2 inhibitor 2 是一种 Cav3.2 T-type Ca2+channels 的抑制剂,-80mV 恒定电位下,其IC50=0.09339 μM。Cav 3.2 inhibitor 2 对小鼠 T 通道依赖性的躯体和内脏疼痛表现出有效的抑制作用。Cav 3.2 inhibitor 2 能够用于研究顽固性疼痛。
T35567 BIX01294 (hydrochloride hydrate)

The methylation of lysine residues on histones plays a central role in determining euchromatin structure and gene expression. The histone methyltransferase (HMTase) G9a can mono- or dimethylate lysine 9 on histone 3 (H3), contributing to early embryogenesis, genomic imprinting, and lymphocyte development. BIX01294 (hydrochloride hydrate) is a selective inhibitor of G9a HMTase (IC50 = 1.7 μM). It less effectively inhibits the HMTase G9a-like protein (GLP; IC50 = 38 μM) and has no effect on other ...
T72388 CBB1007 hydrochloride

CBB1007 hydrochloride,一种可逆的、选择性的高效组蛋白去甲基化酶LSD1的底物竞争性抑制剂,其对hLSD1的IC50值为5.27 uM。
T76014 IGF-I (24-41) (TFA)

IGF-I (24-41) TFA(Insulin-like Growth Factor I (24-41) TFA)是类胰岛素生长因子I的一个氨基酸片段,覆盖24至41位点。作为一种70个氨基酸组成的多肽激素,IGF-I TFA对神经元和神经胶质细胞具有营养作用,而且在调节全身生长激素(GH)活性中扮演关键角色。它还具备合成代谢、抗氧化、抗炎及细胞保护功能,对躯体生长及行为发育调节作用显著。
T72244 CBB1007 trihydrochloride

CBB1007三盐酸盐是 LSD1选择性抑制剂,IC50值为5.27uM。

化合物

Oct3/4-inducer-1
Cat.No: T3221
Synonym: 2-(4-(4-methoxybenzyloxy)phenyl)acetonitrile,2-(4-[(4-甲氧基苄基)氧基]苯基)乙腈
Target: Others, OCT
Moxnidazole
Cat.No: T68110
Synonym:
Target:
Phe-Met-Arg-Phe Like Peptide acetate
Cat.No: TP1057L
Synonym: Pqdpflrfamide acetate,Phe-Met-Arg-Phe Like Peptide acetate(98495-35-3 free base)
Target: Others
MM-102 TFA
Cat.No: T8768
Synonym: HMTase Inhibitor IX TFA
Target: Histone Methyltransferase
RSC-133
Cat.No: T23271
Synonym:
Target: Others
Dynorphin (2-17) (porcine)
Cat.No: T82520
Synonym:
Target:
Phe-Met-Arg-Phe Like Peptide, Snail Helix aspersa
Cat.No: TP1057
Synonym: Phe-Met-Arg-Phe Like Peptide
Target:
CYT296
Cat.No: T78520
Synonym:
Target: Others
Cav 3.2 inhibitor 2
Cat.No: T63606
Synonym:
Target:
BIX01294 (hydrochloride hydrate)
Cat.No: T35567
Synonym:
Target:
CBB1007 hydrochloride
Cat.No: T72388
Synonym:
Target:
IGF-I (24-41) (TFA)
Cat.No: T76014
Synonym:
Target:
CBB1007 trihydrochloride
Cat.No: T72244
Synonym:
Target:
TargetMol Loading
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