Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T28498L |
rac-CCT-250863 HCl
rac-CCT-250863 HCl(1364269-06-6 Free base) |
Apoptosis | Apoptosis |
rac-CCT-250863 HCl 是一种具有选择性和可逆性的 NEK 2 抑制剂。rac-CCT-250863 HCl 能诱导细胞周期停滞,对癌细胞有较好的抗增殖活性,与 Pomalidomide 联用能诱导细胞凋亡,可用于联合抗癌的研究。 | |||
T28498 |
rac-CCT-250863
|
||
Rac-CCT-250863, a potent Nek2 inhibitor, exhibits selectivity for Nek2 over PLK1, MPS1, Cdk2 and Aurora A. |