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Cat. No. Product Name Target Signaling Pathways
T8873 Bractoppin

Others; DNA/RNA Synthesis Cell Cycle/Checkpoint; DNA Damage/DNA Repair; Others
Bractoppin 是一种BRCA1 (t)BRCT domain 识别磷酸肽的选择性抑制剂,IC50为 74 nM。它优先抑制 BRCA1 -tBRCT 依赖的 DNA 损伤。它减少 BRCA1 对 DNA 断裂片段的招募,进而抑制损伤诱导的 G2 期阻滞和重组酶 RAD51 的组装。
TP2211 2B-(SP)

Others Others
Selective phosphopeptide substrate for glycogen synthase kinase-3 (GSK-3)
T41019 Histone H1-derived Peptide

Histone H1-derived Peptide

Histone H1-derived peptide is a phosphopeptide with peptide substrates that consist of a sequence aligned with the optimal recognition motif for cyclin-dependent kinases (CDKs).
T40219 CGP78850

CGP78850 is a potent and selective Grb2 SH2-phosphopeptide interaction antagonist that holds potential for cancer research.
TP2084 N-Acetyl-O-phosphono-Tyr-Glu Dipentylamide

Phosphopeptide; binds to the src SH2 domain.
TP2085 Ac-Tyr(PO3H2)-Glu-Glu-Ile-Glu-OH

N-Acetyl-O-phosphono-Tyr-Glu-Glu-Ile-Glu

Phosphopeptide ligand for the src SH2 domain (IC50 = 1 μM). Blocks src interactions with EGFR and FAK.
T38965 EPQpYEEIPIYL

EPQpYEEIPIYL, a phosphopeptide, is a ligand for the Src homology 2 (SH2) domain. It activates members of the Src family, such as Lck, Hck, and Fyn, through the binding interaction with SH2 domains.
TP2053 Caffeic acid-pYEEIE

Phosphopeptide ligand for the src SH2 domain (IC50 = 42 nM); displays 30-fold higher affinity than N-acetyl-O-phosphono-Tyr-Glu-Glu-Ile-Glu (Ac-pYEEIE,).
T75929 Caffeic acid-pYEEIE TFA

Caffeic acid-pYEEIE TFA 是一种非磷酸肽抑制剂,对 GST-Lck-SH2 结构域具有强大的结合亲和力。

化合物

Bractoppin
Cat.No: T8873
Synonym:
Target: Others, DNA/RNA Synthesis
2B-(SP)
Cat.No: TP2211
Synonym:
Target: Others
Histone H1-derived Peptide
Cat.No: T41019
Synonym: Histone H1-derived Peptide
Target:
CGP78850
Cat.No: T40219
Synonym:
Target:
N-Acetyl-O-phosphono-Tyr-Glu Dipentylamide
Cat.No: TP2084
Synonym:
Target:
Ac-Tyr(PO3H2)-Glu-Glu-Ile-Glu-OH
Cat.No: TP2085
Synonym: N-Acetyl-O-phosphono-Tyr-Glu-Glu-Ile-Glu
Target:
EPQpYEEIPIYL
Cat.No: T38965
Synonym:
Target:
Caffeic acid-pYEEIE
Cat.No: TP2053
Synonym:
Target:
Caffeic acid-pYEEIE TFA
Cat.No: T75929
Synonym:
Target:
TargetMol Loading
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