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抑制剂 & 化合物

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Cat. No. Product Name Target Signaling Pathways
T61850 Adenosine receptor inhibitor 1

Adenosine receptor inhibitor 1 is a highly potent and selective antagonist of adenosine receptor (AR). It exhibits exceptional affinity for A1 AR, A2A AR, A2B AR, and A3 AR, with respective Ki values of >1000, 68.5, >1000, >1000 nM. This compound demonstrates notable antinociceptive, anti-inflammatory, and peripheral analgesic properties. Therefore, Adenosine receptor inhibitor 1 holds great promise for investigating cancer and neurodegenerative diseases [1].

化合物

Adenosine receptor inhibitor 1
Cat.No: T61850
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T7907 7-Methoxyflavone

Others Others
7-Methoxyflavone 是一种分离自 Zornia brasiliensis 的化合物。它能够抑制福尔马林疼痛反应神经源期的舔爪时间 (65.6%),有外周镇痛活性,但不影响炎症期的伤害性反映。

天然产物

7-Methoxyflavone
Cat.No: T7907
Synonym:
Target: Others
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