Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T79800 |
pan-KRAS-IN-2
|
Ras | GPCR/G Protein; MAPK |
Pan-KRAS-IN-2(compound 6)是一种抑制剂,对KRAS WT及其多种突变体(G12D、G12C、G12V、G12S、G12A、Q61H)表现出极高的抑制活性,其IC50均不超过10 nM;然而对KRAS G13D的抑制活性较低,IC50超过10 μM。 |