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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T6956L Protirelin Acetate(24305-27-9 free base)

Thyroliberin Acetate,TRF Acetate,Synthetic thyrotropin-releasing hormone Acetate,Lopremone Acetate,pGlu-His-Pro-NH2 Acetate,TRH Acetate

Thyroid hormone receptor(THR) Endocrinology/Hormones
Protirelin Acetate(24305-27-9 free base) (Thyroliberin Acetate) 是一种三肽,可刺激促甲状腺素和催乳素的释放。
T19511 PGlu-3-methyl-His-Pro-NH2 TFA

A-42872 TFA

Others Others
PGlu-3-methyl-His-Pro-NH2 TFA, enhances binding to pituitary TRH receptors and increases stimulation of thyroid-stimulating hormone (TSH) release from the pituitary.
T82307 Glp-His-Pro-Gly-NH2

pGlu-His-Pro-Gly-NH2

pGlu-His-Pro-Gly-NH2(Glp-His-Pro-Gly-NH2)为含四氨基酸肽类化合物,可激发促性腺激素、黄体生成素(LH)与促卵泡激素(FSH)释放。
T71149 Triptorelin pamoate

Triptorelin, a decapeptide (pGlu-His-Trp-Ser-Tyr-D-Trp-Leu-Arg-Pro-Gly-NH2), is a gonadotropin-releasing hormone agonist (GnRH agonist) used as the acetate or pamoate salts. By causing constant stimulation of the pituitary, it decreases pituitary secretion of gonadotropins luteinizing hormone (LH) and follicle stimulating hormone (FSH). Like other GnRH agonists, triptorelin may be used in the treatment of hormone-responsive cancers such as prostate cancer or breast cancer, precocious puberty, es...

化合物

Protirelin Acetate(24305-27-9 free base)
Cat.No: T6956L
Synonym: Thyroliberin Acetate,TRF Acetate,Synthetic thyrotropin-releasing hormone Acetate,Lopremone Acetate,pGlu-His-Pro-NH2 Acetate,TRH Acetate
Target: Thyroid hormone receptor(THR)
PGlu-3-methyl-His-Pro-NH2 TFA
Cat.No: T19511
Synonym: A-42872 TFA
Target: Others
Glp-His-Pro-Gly-NH2
Cat.No: T82307
Synonym: pGlu-His-Pro-Gly-NH2
Target:
Triptorelin pamoate
Cat.No: T71149
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T6956 Protirelin

Lopremone,pGlu-His-Pro-NH2,Synthetic thyrotropin-releasing hormone,Thyroliberin,TRH,普罗瑞林,TRF

Thyroid hormone receptor(THR); Endogenous Metabolite Endocrinology/Hormones; Metabolism
Protirelin (Thyroliberin) 是高度保守的神经肽,具有促甲状腺激素水平的激素控制作用,及神经调节功能。

天然产物

Protirelin
Cat.No: T6956
Synonym: Lopremone,pGlu-His-Pro-NH2,Synthetic thyrotropin-releasing hormone,Thyroliberin,TRH,普罗瑞林,TRF
Target: Thyroid hormone receptor(THR), Endogenous Metabolite
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