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Targets Recommended: S6 Kinase

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抑制剂 & 化合物

1

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T6878 LJI308

S6 Kinase MAPK; PI3K/Akt/mTOR signaling
LJI308 是泛RSK 抑制剂,对 RSK1、RSK2 和 RSK3 的IC50分别为 6、4 和 13 nM。它抑制辐照、EGF 处理和表达 KRAS 突变的细胞中 RSK (T359/S363) 和 YB-1 (S102) 的磷酸化。

化合物

LJI308
Cat.No: T6878
Synonym:
Target: S6 Kinase
Cat. No. Product Name Species Expression System
TMPY-04392 RSK3 Protein, Human, Recombinant (GST)

HU-2,ribosomal protein S6 kinase, 90kDa, polypeptide 2,S6K-α...

Human Baculovirus Insect Cells
Ribosomal protein S6 kinase alpha-2, also known as 9 kDa ribosomal protein S6 kinase 2, MAP kinase-activated protein kinase 1c, MAPK-activated protein kinase 1c, Ribosomal S6 kinase 3, RSK-3, RPS6KA2 and MAPKAPK1C, is a nucleus protein that belongs to the protein kinase superfamily, AGC Ser/Thr protein kinase family and S6 kinase subfamily. RPS6KA2 / RSK-3 is expressed in many tissues. Highest expression is in lung and skeletal muscle. The expression of RPS6KA2 reduced proliferation, caused G1 a...

重组蛋白

RSK3 Protein, Human, Recombinant (GST)
Cat.No: TMPY-04392
Species: Human
Expression System: Baculovirus Insect Cells
TargetMol Loading
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