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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T60199 NCRW0005-F05

GPR Endocrinology/Hormones; GPCR/G Protein
NCRW0005-F05 是一种有效的孤儿 G 蛋白偶联受体GPR139的激动剂,IC50为 0.21 μM。NCRW0005-F05 可用于研究糖尿病、肥胖症和帕金森的研究。
TP1982L Neuropeptide S (Rat) acetate

Neuropeptide Y Receptor GPCR/G Protein; Neuroscience
Neuropeptide S (Rat) acetate 是以前孤儿 G 蛋白偶联受体的内源性配体,现在称为 NPS 受体。它可用于神经系统疾病的研究。
T0755 Carglumic Acid

Carbaglu,N-Carbamylglutamate,N-Carbamyl-L-glutamic acid,氨甲酰谷氨酸,Carbamylglutamic acid,Carbamino-L-glutamic acid,Ureidoglutaric acid

Others Others
Carglumic Acid (Ureidoglutaric acid) 是一种 N-乙酰谷氨酸 (NAG) 的功能类似物和氨甲酰磷酸合成酶 1(CPS1)的活化剂,可用于与 N-乙酰谷氨酸合成酶 (NAGS) 缺陷相关的急性和慢性高氨血症的研究。
T73545 TH470

TH470 是一种高选择性的LIMK1/2(LIM 激酶 1/2) 抑制剂 (LIMK1IC50=9.8 nM ; LIMK2IC50=13 nM),可用于孤儿病的研究。
T37187 D-erythro/L-threo Lysosphingomyelin (d18:1)

D-erythro/L-threo Lysosphingomyelin (d18:1)

Lysosphingomyelin is an endogenous bioactive sphingolipid and a constituent of lipoproteins.1,2It is produced by the removal of the acyl group from sphingomyelin by a deacylase and acts as a precursor in the biosynthesis of sphingosine-1-phosphate . D-erythroLysosphingomyelin is an agonist of the S1P receptors S1P1, S1P2, and S1P3(EC50s = 167.7, 368.1, and 482.6 nM, respectively, for the human receptors).3It is also an agonist of the orphan receptor ovarian cancer G protein-coupled receptor 1 (O...

化合物

NCRW0005-F05
Cat.No: T60199
Synonym:
Target: GPR
Neuropeptide S (Rat) acetate
Cat.No: TP1982L
Synonym:
Target: Neuropeptide Y Receptor
Carglumic Acid
Cat.No: T0755
Synonym: Carbaglu,N-Carbamylglutamate,N-Carbamyl-L-glutamic acid,氨甲酰谷氨酸,Carbamylglutamic acid,Carbamino-L-glutamic acid,Ureidoglutaric acid
Target: Others
TH470
Cat.No: T73545
Synonym:
Target:
D-erythro/L-threo Lysosphingomyelin (d18:1)
Cat.No: T37187
Synonym: D-erythro/L-threo Lysosphingomyelin (d18:1)
Target:
Cat. No. Product Name Target Signaling Pathways
TN6715 7-Ketocholesterol

Others Others
7-Ketocholesterol 是胆固醇的代谢物。

天然产物

7-Ketocholesterol
Cat.No: TN6715
Synonym:
Target: Others
TargetMol Loading
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