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Cat. No. Product Name Target Signaling Pathways
T22371 Mivacurium dichloride

米库氯铵,Mivacurium chloride,二氯美维库铵

AChR Neuroscience
Mivacurium dichloride (Mivacurium chloride) 是苄基异喹啉衍生物,可与 nAChR 偶联,以减少或抑制乙酰胆碱对肌肉细胞末端盘的去极化作用。它也是非去极化短效的神经肌肉阻滞剂和骨骼肌松弛剂。
T6397 Atracurium besylate

Tracrium,51W89,BW-33A,苯磺酸阿曲库铵

AChR Neuroscience
Atracurium besylate (51W89) 是一种神经肌肉阻断剂,ED95为0.2 mg/kg。
T1594 Vecuronium bromide

ORG NC 45,维库溴铵

AChR Neuroscience
Vecuronium bromide (ORG NC 45) 是一种合成的中效单季铵盐类固醇和非去极化神经肌肉阻滞剂,具有肌肉松弛活性。
T0156 Rocuronium bromide

ORG 9426,罗库溴铵,ORG 9426 (Bromide)

AChR Neuroscience
Rocuronium bromide (ORG 9426) 是一种氨基甾体类的、非去极化的神经肌肉受体抑制剂,也是一种肌肉松弛剂。
T12748 Rocuronium

罗库铵,Org-9426

Others Others
Rocuronium is an blocker of aminosteroid non-depolarizing neuromuscular.
T29846 Alcuronium free base

Alcuronium,Alcuronum,Diallylnortoxiferine,Alcuronium kation,Alloferine

Alcuronium free base is a non-depolarizing skeletal muscle relaxant similar to Tubocurarine. It is used as an anesthesia adjuvant.
T25636 Laudexium

Laudexium ion,Laudexium cation

Laudexium is a neuromuscular blocking drug or skeletal muscle relaxant in the category of non-depolarizing neuromuscular-blocking drugs. It is used adjunctively in surgical anesthesia to facilitate endotracheal intubation and to provide skeletal muscle re
T33638 Neostigmine Iodide

SB 24,SB24,TL1321,TL 1321,TL-1321,SB-24

Neostigmine Iodide is a parasympathic compound used as a reversible acetylcholinesterase inhibitor to improve muscle tone in patients with myasthenia gravis and in routine anesthesia to reverse the effects of non-depolarizing muscle relaxants such as rocu
T70269 Hexamethonium chloride dihydrate

Hexamethonium chloride dihydrate is a non-depolarizing NMJ blocker and nAChR antagonist. It has previously been used to treat hypertension. It inhibits sympathetic nervous system activity and acts as a skeletal muscle relaxant.
T68645 Hexamethonium monotartrate

Hexamethonium monotartrate is a non-depolarizing NMJ blocker and nAChR antagonist. It has previously been used to treat hypertension. It inhibits sympathetic nervous system activity and acts as a skeletal muscle relaxant.
T69161 Hexamethonium bromide dihydrate

Hexamethonium bromide dihydrate is a non-depolarizing NMJ blocker and nAChR antagonist. It has previously been used to treat hypertension. It inhibits sympathetic nervous system activity and acts as a skeletal muscle relaxant.
T68811 Trimetaphan camsilate

Trimetaphan camsilate is a drug that counteracts cholinergic transmission at the ganglion type of nicotinic receptors of the autonomic ganglia and therefore blocks both the sympathetic nervous system and the parasympathetic nervous system. It acts as a non-depolarizing competitive antagonist at the nicotinic acetylcholine receptor, is short-acting, and is given intravenously.
T75283 Atracurium

Atracurium (BW-33A free acid)为高效的竞争性非去极化神经肌肉阻滞剂,兼具AChR受体拮抗作用。该化合物能够诱导支气管收缩及实现神经肌肉阻滞,并促进星形胶质细胞分化[5]。
T37702 Pancuronium (bromide hydrate)

Pancuronium is an aminosteroid antagonist of muscle-type nicotinic acetylcholine receptors (nAChRs) with an IC50value of 14.8 nM using patch clamp electrophysiology in BOSC23 cells expressing mouse nAChRs.1It acts as a non-depolarizing neuromuscular blocking agent.2Pancuronium enhances anesthesia induced by isoflurane , reducing immobilization with an ED50value of 1.62 μg/kg.3 1.Liu, M., and Dilger, J.P.Site selectivity of competitive antagonists for the mouse adult muscle nicotinic acetylcholin...

化合物

Mivacurium dichloride
Cat.No: T22371
Synonym: 米库氯铵,Mivacurium chloride,二氯美维库铵
Target: AChR
Atracurium besylate
Cat.No: T6397
Synonym: Tracrium,51W89,BW-33A,苯磺酸阿曲库铵
Target: AChR
Vecuronium bromide
Cat.No: T1594
Synonym: ORG NC 45,维库溴铵
Target: AChR
Rocuronium bromide
Cat.No: T0156
Synonym: ORG 9426,罗库溴铵,ORG 9426 (Bromide)
Target: AChR
Rocuronium
Cat.No: T12748
Synonym: 罗库铵,Org-9426
Target: Others
Alcuronium free base
Cat.No: T29846
Synonym: Alcuronium,Alcuronum,Diallylnortoxiferine,Alcuronium kation,Alloferine
Target:
Laudexium
Cat.No: T25636
Synonym: Laudexium ion,Laudexium cation
Target:
Neostigmine Iodide
Cat.No: T33638
Synonym: SB 24,SB24,TL1321,TL 1321,TL-1321,SB-24
Target:
Hexamethonium chloride dihydrate
Cat.No: T70269
Synonym:
Target:
Hexamethonium monotartrate
Cat.No: T68645
Synonym:
Target:
Hexamethonium bromide dihydrate
Cat.No: T69161
Synonym:
Target:
Trimetaphan camsilate
Cat.No: T68811
Synonym:
Target:
Atracurium
Cat.No: T75283
Synonym:
Target:
Pancuronium (bromide hydrate)
Cat.No: T37702
Synonym:
Target:
TargetMol Loading
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