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抑制剂 & 化合物

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Cat. No.	Product Name	Target	Signaling Pathways
TP1363L	Neurokinin B acetate(86933-75-7 free base) 神经激肽 B醋酸盐,Neurokinin K	Neurokinin receptor	GPCR/G Protein; Neuroscience
	Neurokinin B acetate(86933-75-7 free base) 是属于速激肽家族的神经激肽 B 的醋酸盐形式。神经激肽与神经激肽受体 1 (NK1R)、nk2r 和 NK3R 结合，并介导其生物学效应。
TP1363	Neurokinin B
	Neurokinin B (NKB) belongs in the family of tachykinin peptides. Neurokinin B is implicated in a variety of human functions and pathways such as the secretion of gonadotropin-releasing hormone.
TP1279	Neurokinin B (TFA) 神经激肽 B 三氟乙酸盐,Neurokinin B TFA
	Neurokinin B TFA belongs to the tachykinin family.Neurokinin B binds to a series of GPCR, including neurokinin receptors 1 (NK1R), NK2R, and nk3r, to modulate their biological effects
T16849	SB-222200	Neurokinin receptor	GPCR/G Protein; Neuroscience
	SB-222200 是一种选择性口服活性的，具有血脑屏障渗透性的 NK-3 受体拮抗剂，用于中枢神经系统疾病的研究。
T80914	Tyr0-Neurokinin B Tyr-NKB
	Tyr0-Neurokinin B (Tyr-NKB)为Neurokinin B的类似物，具有引发膀胱收缩的生物活性。
T76436	[MePhe7]-Neurokinin B
	[MePhe7]-Neurokinin B为NK-3受体(NK3R)激动剂，具有3 nM的IC50值。通过激活神经激肽3受体，[MePhe7]-Neurokinin B能够调节脉冲促性腺激素释放激素(GnRH)的分泌，成为调控该过程的潜在调节剂。
T76427	(D-Pro2,D-Trp6,8,Nle10)-Neurokinin B
	(D-Pro2,D-Trp6,8,Nle10)-Neurokinin B 是 Neurokinin B(Neurokinin Receptor) 的竞争性拮抗剂，pA2 为 5.5，对 Substance P 或 Neurokinin A 没有影响。
T24285	L 363851 L363851,L-363851,L363,851,L 363,851,L-363,851
	L 363851 is a neurokinin B agonist.
T76431	GR 83074
	GR 83074 是一种有效的选择性 NK-2(Neurokinin Receptor) 拮抗剂，pKB 为 8.23。GR 83074 对 NK-3 没有活性，并表现出 340 倍的 NK-2/NK-1 选择性。
T38276	Benzomalvin C
	Benzomalvin C is a weak antagonist of the neurokinin-1 (NK1) receptor inhibiting binding of substance P by 46% when used at 100 μg/ml in vitro. It is also a weak inhibitor of indolamine 2,3-dioxygenase (IDO) with an IC50 value of 130 μM for recombinant IDO. It was isolated from Penicillium and contains an epoxide group at C-19 and C-20, which is not present in benzomalvins A, B, or E.
T36053	D-Lysine lactam
	D-Lysine lactam is a chiral building block.1,2It has been used in the synthesis of a chiral antibiotic synthetic intermediate, as well as in the stereoselective synthesis of neurokinin (NK) receptor antagonists. 1.Kumar, A., Bhashkar, B., Bhavsar, J., et al.Catalytic reduction: Efficient synthesis of chiral key intermediate of besifloxacin hydrochlorideDer Pharma Chemica7(9)297-3000(2015) 2.Gerspacher, M., Lewis, C., Ball, H.A., et al.Stereoselective preparation of N-[(R,R)-(E)-1-(3,4-dichlorobe...
T32007	GSK256471 GSK 256471,GSK-256471
	GSK256471 is a potent selective NK(3) antagonist that shows a high affinity for recombinant human (PK (I) value 8.9) and native guinea pig (PK (I) value 8.4) tachykinin NK(3) receptors. In vitro functional assessment showed that GSK256471 reduced the E(Ma

化合物

Neurokinin B acetate(86933-75-7 free base)

Cat.No: TP1363L

Synonym: 神经激肽 B醋酸盐,Neurokinin K

Target: Neurokinin receptor

Cat.No: TP1363

Neurokinin B (TFA)

Cat.No: TP1279

Synonym: 神经激肽 B 三氟乙酸盐,Neurokinin B TFA

Cat.No: T16849

Target: Neurokinin receptor

Tyr0-Neurokinin B

Cat.No: T80914

Synonym: Tyr-NKB

[MePhe7]-Neurokinin B

Cat.No: T76436

(D-Pro2,D-Trp6,8,Nle10)-Neurokinin B

Cat.No: T76427

Cat.No: T24285

Synonym: L363851,L-363851,L363,851,L 363,851,L-363,851

Cat.No: T76431

Cat.No: T38276

D-Lysine lactam

Cat.No: T36053

Cat.No: T32007

Synonym: GSK 256471,GSK-256471

Cat. No.	Product Name	Target	Signaling Pathways
T38033	Benzomalvin B
	Benzomalvin B is a fungal metabolite originally isolated from Penicillium. It acts as an antagonist of neurokinin-1 (NK1) receptors, inhibiting binding of substance P by 24% in vitro when used at a concentration of 100 μg/ml.

天然产物

Cat.No: T38033

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