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Cat. No. Product Name Target Signaling Pathways
T0203 Sumatriptan succinate

舒马普坦琥珀酸盐,GR 43175,琥珀酸舒马曲坦

5-HT Receptor GPCR/G Protein; Neuroscience
Sumatriptan succinate (GR 43175) 是一种5-HT1受体激动剂,可作用于偏头疼的急性治疗。
T26079 RI 61

RI-61,Pro-his-pro-phe-his-leu-phe-val-phe,RI61

RI 61 (sumatriptan succinate) is utilized in the therapy of migraine, cluster headaches, new daily persistent headache, and cyclic vomiting syndrome.
T60345 Frovatriptan

Frovatriptan is a highly potent agonist of the 5-HT 1B//D receptors, exhibiting the highest potency among triptan compounds. It possesses prominent cerebroselectivity. Frovatriptan demonstrates efficacy and even superiority in certain endpoints, including when administered during the headache phase of migraine attacks accompanied by aura [1].
T60989 Sumatriptan hydrochloride

Sumatriptan (GR 43175) hydrochloride 可用于研究偏头痛,它是一种口服有效的5-HT1受体激动剂。Sumatriptan hydrochloride 对5-HT1D、5-HT1B 和5-HT1A 受体的 Ki 值分别为 17 nM、27 nM 和 100 nM。

化合物

Sumatriptan succinate
Cat.No: T0203
Synonym: 舒马普坦琥珀酸盐,GR 43175,琥珀酸舒马曲坦
Target: 5-HT Receptor
RI 61
Cat.No: T26079
Synonym: RI-61,Pro-his-pro-phe-his-leu-phe-val-phe,RI61
Target:
Frovatriptan
Cat.No: T60345
Synonym:
Target:
Sumatriptan hydrochloride
Cat.No: T60989
Synonym:
Target:
TargetMol Loading
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