Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T80495 |
mHuwentoxin-IV
|
Sodium Channel | Membrane transporter/Ion channel |
mHuwentoxin-IV是一种经天然修饰的Huwentoxin-IV。该化合物针对背根神经节中河豚毒素敏感(TTX-S)电压门控钠通道(sodium channels)表现出抑制作用,IC50值为54.16 nM。mHuwentoxin-IV对这些钠通道的抑制作用并不会因强去极化电压而逆转。 |