Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T60745 |
hCAIX-IN-5
|
Carbonic Anhydrase | Metabolism |
hCAIX-IN-5 是一种具有选择性的 hCAIX 抑制剂,对 hCAI, hCAII,hCAIV,hCAIX 的 有抑制作用, Ki值分别为 >10000, >10000, 130.7, 829.1 nM。 | |||
T60602 | hCAIX/XII-IN-5 | ||
hCAIX/XII-IN-5 (Coumarin 9a) 是一种碳酸酐酶 (CA) 抑制剂,具有出色的 hCA IX/XII 选择性,对 hCA I 和 hCA II 的Ki 值分别为 93.9 和 85.7 nM。hCAIX/XII-IN-5 对癌细胞具有抗增殖活性,可延迟细胞周期并诱导细胞凋亡。 | |||
T61769 | hCAXII-IN-5 | ||
hCAXII-IN-5 (compound 6o) is a highly effective and specific inhibitor of hCAXII. The compound exhibits impressive binding affinities, with Ki values of >10000, >10000, 286.1, and 1.0 nM for hCAI, hCAII, hCAIX, and hCAXII, respectively [1]. |