Cat. No. | Product Name | Target | Signaling Pathways |
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T63631 |
hCAII-IN-2
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hCAII-IN-2 是胞质型人碳酸酐酶 (hCA) 抑制剂,能够作用于 hCA I (Ki: 261.4 nM)、hCA II (Ki: 3.8 nM)、hCA IX (Ki: 19.6 nM)和 hCA XII (Ki: 45.2 nM)。 | |||
T63789 | β-Glucuronidase/hCAII-IN-2 | ||
β-Glucuronidase/hCAII-IN-2 是 β-glucuronidase 和 hCA II 的有效抑制剂,他们的IC50值分别为 670.7 μM 和 21.77 μM。 | |||
T63805 |
β-Glucuronidase/hCAII-IN-1
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β-Glucuronidase/hCAII-IN-2 (Compound 12e) 是一种有效的β-glucuronidase 和 hCA II 抑制剂,其 IC50分别为 440.1 μM 和 4.91 μM。 | |||
T61015 |
hCAIX/XII-IN-2
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hCAIX/XII-IN-2 (compound 6a) 是有效的 hCAIX 和 hCAXII 的选择性抑制剂,其对于hCAI、hCAII、hCAIX 和 hCAXII 的Ki 值分别为 >10000、>10000、30.0、3.6 nM。 | |||
T61164 | hCAII-IN-3 | ||
hCAII-IN-3 (Compound 16) is an inhibitor of human carbonic anhydrase (hCA). It exhibits high affinity for hCA I, hCA II, hCA IX, and hCA XII, with Ki values of 403.8 nM, 5.1 nM, 10.2 nM, and 5.2 nM, respectively. Notably, hCA IX-IN-2 demonstrates anticancer activity [1]. |