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Cat. No. | Product Name | Target | Signaling Pathways |
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T3124 |
Carbendazim
Bavistin,Carbendazole,多菌灵,Mercarzole |
Antifungal | Microbiology/Virology |
Carbendazim (Mercarzole) 是一种具有抗肿瘤活性的苯并咪唑衍生物,可用于癌症研究。它是一种口服广谱苯并咪唑杀菌剂,可作为真菌疾病研究的杀虫剂。 | |||
T70267 |
ADL 08-0011 HCl
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ADL 08-0011 is an active metabolite of the μ-opioid receptor antagonist alvimopan. It is produced from alvimopan via amide hydrolysis by gut microbiota. ADL 08-0011 is a μ-opioid receptor antagonist (Ki = 0.25 nM). It is selective for μ-opioid receptors over κ- and δ-opioid receptors (Kis = 15.8 and 31.6 nM, respectively). ADL 08-0011 inhibits endomorphin 1-induced inhibition of electrically induced contraction of isolated guinea pig ileum (pA2 = 9.4). In vivo, ADL 08-0011 (0.03-1 mg/kg) reverse... |
Cat. No. | Product Name | Target | Signaling Pathways |
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T4S0554 |
Theaflavine-3,3'-digallate
TFBG,theaflavin digallate,3,3’-二没食子酸酯茶黄素 |
Others | Others |
Theaflavine-3,3'-digallate (theaflavin digallate) 和乳酸一起可以减少单纯疱疹病毒的传播。 | |||
T8878 |
urolithin M6
尿石素M6,3,8,9,10-tetrahydroxy urolithin |
Others | Others |
urolithin M6 (3,8,9,10-tetrahydroxy urolithin) 是一种由肠道微生物群产生的鞣花单宁代谢物,被确定为推定的没食子黄素模拟物。 | |||
T3840 |
Dihydroresveratrol
3,4',5-Trihydroxybibenzyl,二氢白藜芦醇,二氢藜芦醇 |
Estrogen Receptor/ERR; Others | Endocrinology/Hormones; Others |
Dihydroresveratrol (3,4',5-Trihydroxybibenzyl) 是一种激素受体调节剂,是一种植物雌激素。它在皮摩尔和纳摩尔浓度下促进前列腺和乳腺癌细胞增殖。 | |||
TN6733 |
Kansuiphorin C
KPC,甘遂大戟萜酯C |
Others | Others |
Kansuiphorin C (KPC) 是一种具有多种生物活性的天然产物。它能够调节肠道菌群及相关代谢功能,并可以改善恶性腹水。 | |||
T2A2428 |
2-Hydroxy-4-methoxybenzoic acid
2-Hydroxy-p-anisic Acid,4-Methoxysalicylic acid,对甲氧基水杨酸,2-羟基-4-甲氧基苯甲酸 |
Others | Others |
2-Hydroxy-4-methoxybenzoic acid (2-Hydroxy-p-anisic Acid) 是一种甲氧基苯甲酸的衍生物,它是一种潜在的生物标志物。 | |||
T3737 |
3-(2,4-Dihydroxyphenyl)propanoic acid
3-(2,4-二羟基苯)丙酸,Hydroumbellic acid,2,4-Dihydroxyhydrocinnamic acid |
Tyrosinase | Proteases/Proteasome |
3-(2,4-Dihydroxyphenyl)propanoic acid (Hydroumbellic acid) 是竞争性酪氨酸酶 (tyrosinase) 抑制剂,可抑制 L-Tyrosine 和 DL-DOPA,IC50和 Ki 分别为 3.02 μM 和 11.5 μM。 | |||
T37404 |
O-Desmethylangolensin
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O-Desmethylangolensin is a gut microbiota metabolite of daidzein, a soy isoflavone. It demonstrates antioxidant activity[1][2]. | |||
T77988 |
Phenyl sulfate
Phenyl hydrogen sulfate |
Endogenous Metabolite | Metabolism |
Phenyl sulfate为肠道微生物衍生的口服活性代谢物,能在糖尿病实验模型中诱发蛋白尿及足细胞损伤,其可能成为糖尿病肾病的疾病标志物和未来治疗靶点。 | |||
T83804 |
5-(3'-Hydroxyphenyl)-γ-Valerolactone
(3’-hydroxy)-PVL,δ-(3’-Hydroxyphenyl)-γ-VL,5-(3’-Hydroxyphenyl)-γ-VL,δ-(3’-Hydroxyphenyl)-γ-Valerolactone |
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5-(3'-羟基苯基)-γ-戊内酯是多种多酚的代谢产物,包括(+)-儿茶素和(−)-表儿茶素。这种化合物由肠道微生物从这些多酚中形成。 | |||
T83673 |
4-Hydroxyphenylpropionylglycine
Phloretylglycine,4-hydroxy PPG,Phloretic Acid Glycine Conjugate |
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4-Hydroxyphenylpropionylglycine是一种由条件必需氨基酸酪氨酸代谢形成的代谢产物。通过芳香族氨基酸转氨酶、酪氨酸转氨酶以及肠道微生物作用后,结合甘氨酸共轭生成。此外,4-Hydroxyphenylpropionylglycine也是酚类化合物phloretin的代谢产物。 |