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抑制剂 & 化合物

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天然产物

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Cat. No. Product Name Target Signaling Pathways
T32196 Isariin B

Isariin B is a new cyclodepsipeptide isolated from the entomopathogenic fungus Beauveria felina.
T32195 Isariin

NSC 135015,Isariin D,Isariin C,Isariin B,NSC-135015

Isariin is a cyclodepsipeptide isolated from the fungus Isaria felina.

化合物

Isariin B
Cat.No: T32196
Synonym:
Target:
Isariin
Cat.No: T32195
Synonym: NSC 135015,Isariin D,Isariin C,Isariin B,NSC-135015
Target:
Cat. No. Product Name Target Signaling Pathways
TCS1554 trans-Benzylideneacetone

反式苯亚甲基丙酮,Acetocinnamone,亚苄基丙酮

Phospholipase Metabolism
trans-Benzylideneacetone (Acetocinnamone) 是一种革兰氏阴性致病性线虫细菌嗜线虫(Xenorhabdus nematophila) 的代谢产物,是一种针对磷脂酶 A2 (PLA2) 的酶抑制剂,也是一种免疫抑制剂。
T38016 Hirsutide

Hirsutide is a cyclotetrapeptide fungal metabolite produced by the entomopathogenic fungus Hirsutella. It has antibacterial activity against C. pyogenes, S. aureus, P. aeruginosa, and K. pneumonia (MICs = 25, 13, 6, and 21 μg/cm3, respectively). Hirsutide also has antifungal activity against C. albicans, M. audouinii, A. niger, and Ganoderma (MICs = 13, 6, 25, and 6 μg/cm3, respectively).
T38262 Sphingosine (d14:1)

Sphingosine (d14:1) is a bioactive sphingolipid that has been found in B. mori (silkworm), P. clarkii (crayfish), and A. aurita (jellyfish) extracts. It increases the germination rate of N. rileyi, an entomopathogenic fungus, with an EC50 value of 10.2 nM. Sphingosine (d14:1) inhibits protein kinase C (PKC) in vitro (IC50 = 7.3 mol%) as well as superoxide generation induced by phorbol 12-myristate 13-acetate in neutrophils and reduces growth of CHO cells (IC50s = 19 and 8 μM, respectively).

天然产物

trans-Benzylideneacetone
Cat.No: TCS1554
Synonym: 反式苯亚甲基丙酮,Acetocinnamone,亚苄基丙酮
Target: Phospholipase
Hirsutide
Cat.No: T38016
Synonym:
Target:
Sphingosine (d14:1)
Cat.No: T38262
Synonym:
Target:
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